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filingDate 2005-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2008-02-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008504296-A
titleOfInvention Novel indazole carboxamide and use thereof
abstract The present invention is directed to novel indazole carboxamide derivatives. In particular, the present invention provides compounds of formula (I) [Wherein R1 and Z are as described herein] And the pharmaceutically acceptable salts thereof. The compounds of the present invention are inhibitors of IKK2 and are useful in the treatment of disorders associated with inappropriate IKK2 (also referred to as IKKβ) activity, such as rheumatoid arthritis, asthma and COPD (chronic obstructive pulmonary disease). Accordingly, the present invention is further directed to pharmaceutical compositions comprising the compounds of the present invention. The present invention is still further directed to methods of inhibiting IKK2 activity and related disorders thereof using a compound of the invention or a pharmaceutical composition comprising a compound of the invention.
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http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2014038623-A1
priorityDate 2004-06-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2734378
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID395196
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ60680
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ71WU4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9638
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2FRW1
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414865594
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8Y2D1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID11668946
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2736256
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3N5K9
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9845
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2AGU8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO49564
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2SC97
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID444556
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421136784
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP49113
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB6CKP4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID17754027
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8XLN7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2S6C4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID62365
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2733699
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ1PDW3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68626860
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID120273
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID5460308
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LMT9
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID416184335
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA5VIG4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID87169756
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LMP1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7YRB5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2RIT6
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1452446
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ54TR5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LMN8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO73909
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2MH06
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2I9L5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LMN7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA0A0R4IYF1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2RFS6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ0BBR3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LMN6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5E5S1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ54P00
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LK35
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP15208
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419514433
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8MKH0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LDT0
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10451
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB9DJN0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LDS6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10450
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ54IH6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LDQ3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCF1MWT5
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID16337
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415753100
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID451544447
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LDN1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3839223
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA6LTA6
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID82408
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LDM5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB8ZKX2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6NSR3
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID7369
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ54DK4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419517633
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6NQ87
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID450673
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ04JT7
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID13728
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9M8S2
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9M342
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415775537
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419508720
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95KV1
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2734619
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3CP33
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60702
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5D7Q0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60701
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9M0X5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP60700
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9M0G5
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419656506
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9M092
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA9AEZ6
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LZU4
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID392871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID453492542
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCC5CJ68
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5WDH1
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LZM4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ042D2
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID114461
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ55G83
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9LX66
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID448485711
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID13399
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID413985283
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415730448
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID281073
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ95181
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ55EU4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ6V919
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8TUS5

Total number of triples: 1048.