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filingDate 2005-06-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2008-01-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008502788-A
titleOfInvention Preparation of polymer conjugates by four-component condensation reaction
abstract Polymer-biomolecule conjugates are generally prepared in a site-specific or site-selective manner by a four-component condensation reaction. This method can be used to prepare conjugates in which two polymer molecules are attached to a single site on a biomolecule. These conjugates are typically water soluble and have advantageous pharmacological properties (eg, reduced immunogenicity and increased circulation time).
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