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filingDate 2007-06-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9da3ce6d97d20ca4d8b0f3dc194d10d8
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publicationDate 2008-05-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2008110960-A
titleOfInvention 6- (Heterocyclic substituted benzyl) -4-oxoquinoline compounds and their use as HIV integrase inhibitors
abstract The following general formula [I] [Wherein each symbol is as described in the specification. Or a pharmaceutically acceptable salt thereof, or a solvate thereof, and a pharmaceutical composition, an anti-HIV agent, and an HIV integrase inhibitor containing the compound. [Effect] The compound of the present invention has an action of inhibiting HIV integrase activity, and is useful as an anti-HIV agent or a therapeutic or preventive agent for AIDS. Moreover, it can become a more effective anti-HIV agent by using together with other anti-HIV agents such as protease inhibitors and reverse transcriptase inhibitors. In addition, having high inhibitory activity specific to integrase can be a safe drug with few side effects for the human body. [Selection figure] None
priorityDate 2006-06-23-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 864.