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filingDate 2004-12-15-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2007-06-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2007514742-A
titleOfInvention Novel 5,6-dihydropyridin-2-one compounds useful as thrombin inhibitors
abstract Compounds of formula (I) (wherein R 1 , R 2a , R 2b , R 3a , R 3b , R 4 , R 5 , R 6 , A, G and L have the meanings indicated in the specification) I will provide a. These compounds are useful as competitive inhibitors of trypsin-like proteases such as thrombin, or are useful as prodrugs thereof, and therefore are particularly useful in situations where inhibition of thrombin is beneficial (for example, where thrombin inhibition is necessary or desirable), For example, it is useful for the treatment of embolism and / or conditions where anticoagulant therapy is applied.
priorityDate 2003-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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Total number of triples: 428.