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filingDate 2004-11-24-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2007-05-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2007512351-A
titleOfInvention GlycoPEGylated erythropoietin
abstract The present invention provides a conjugate between erythropoietin and a PEG moiety. This conjugate is linked via an intact glycosyl linking group interposed between and covalently attached to the peptide and the modifying group. Conjugates are formed from glycosylated peptides by the action of glycosyltransferases. Glycosyltransferases ligate modified sugar moieties onto glycosyl residues on the peptide. Also provided are methods for preparing the conjugates, methods for treating various pathological health conditions with the conjugates, and pharmaceutical formulations containing the conjugates.
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Total number of triples: 1528.