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filingDate 2004-09-02-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2007-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2007505040-A
titleOfInvention Preparation method of water-soluble diterpene and its application
abstract Using an appropriately substituted cyclodextrin as a solubilizer, an aqueous solution of diterpenes such as forskolin, its homologues, analogs and derivatives is prepared to a concentration of about 6%. In the absence of cyclodextrin, some diterpenes, such as forskolin, dissolve only in water to a concentration of about 0.001%. As a preparation for pharmaceutical, cosmetic, nutritional supplements containing diterpenes such as forskolin and homologous substances, topical and systemic applications of such aqueous solutions are found.
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