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filingDate 2004-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2007-03-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2007505039-A
titleOfInvention Improved delivery by hydrophobic modification of easily denatured drugs
abstract Drug formulations that enhance local delivery of drugs to cells are described. A method for reversibly increasing the hydrophobicity of a drug by hydrolytically degrading addition of a hydrophobic site and a method for delivering a modified drug to cells are described. Hydrophobic modifications enhance drug delivery, while facile denaturation minimizes drug entry into untargeted cells.
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