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filingDate 2003-12-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2006-06-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2006515851-A
titleOfInvention Piperidine derivatives useful as CCR5 antagonists
abstract The present invention provides a compound of formula (I) or a pharmaceutically acceptable salt or solvate thereof, wherein the various moieties are as defined in the specification. The present invention also provides pharmaceutical compositions containing the compounds of the present invention and methods of treatment using the compounds of the present invention. The invention also relates to the use of a combination of a compound of the invention and one or more antiviral agents or other agents useful in the treatment of human immunodeficiency virus (HIV). The present invention further includes solid organ transplant rejection, graft-versus-host disease, arthritis, rheumatoid arthritis, inflammatory bowel disease, atopic dermatitis, psoriasis, asthma, allergy or multiple, alone or in combination with other drugs. It also relates to the use of the compounds of the invention in the treatment of sclerosis. Embedded image
priorityDate 2002-12-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22301
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP61815
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP37997
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ29055
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID473183
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410129964
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID415749611
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21329
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID1461021
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426185352
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456373055
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8LKW0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO14746
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID24481
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ2PE73
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP70499
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO97798
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP46651
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DV89
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7JFM4
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504895
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9NBX4
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DV86
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID464372
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DV94
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID2760919
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456371022
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419567920
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21328
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID60871
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID458392451
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID414372168
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419517945
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID457493614
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID456171974
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID135398739
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID72180
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID12721
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID425154543
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504556
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA2T6Z6
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410479690
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DV59

Total number of triples: 352.