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filingDate 2003-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2006-01-05-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2006500422-A
titleOfInvention Lipophilic diesters of chelating agents for inhibiting enzyme activity
abstract The present invention relates to the chelating agent 1,2-bis (2aminophenoxy) ethane-N, N, N ′, N′-tetraacetic acid (BAPTA) for inhibiting the proteolytic activity of certain metalloproteinases and calpains. To the use of a lipophilic diester. The invention further relates to a disease associated with MMP and calpain in a mammal, comprising administering to the mammal in need thereof a pharmaceutical composition comprising a therapeutically effective amount of the lipophilic diester of the chelating agent BAPTA. The present invention relates to a method for preventing, treating or managing a disorder.
priorityDate 2002-09-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID460916
http://rdf.ncbi.nlm.nih.gov/pubchem/anatomy/ANATOMYID5476
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419524027

Total number of triples: 309.