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classificationIPCInventive http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K9-50
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K47-38
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filingDate 2005-02-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c237810b3a91f7a8b960ec60cfc7a843
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publicationDate 2006-09-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2006232789-A
titleOfInvention Composition for oral preparation and method for producing the same
abstract PROBLEM TO BE SOLVED: To provide a composition for oral preparation which can mask an unpleasant taste such as a bitter taste even if it contains a macrolide antibiotic and has a high dissolution property of medicinal ingredients and a method for producing the same. In a composition for oral preparation, a powdered granular composition composed of at least a macrolide antibiotic is coated with a polymer composition composed of a pH-independent water-insoluble polymer and a gastric polymer. The ratio (weight ratio) between the pH-independent water-insoluble polymer and the gastric soluble polymer is adjusted to pH-independent water-insoluble polymer / gastric soluble polymer = 1/1 to 1/20. The pH-independent water-insoluble polymer may be, for example, a cellulose derivative (for example, ethyl cellulose) or a (meth) acrylic polymer. The macrolide antibiotic may be, for example, a 14-membered ring compound such as clarithromycin. [Selection figure] None
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