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filingDate 2002-10-18-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2005-03-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2005506351-A
titleOfInvention Polymer conjugate opioid antagonist
abstract The present invention provides a polymer conjugate of an opioid antagonist, which contains a polymer (eg, poly (ethylene glycol)) covalently attached to the opioid antagonist. The linkage between the polymer and the opioid antagonist is preferably hydrolytically stable. The present invention also includes a method of treating one or more side effects (eg, constipation, nausea or pruritus) associated with the use of an opioid antagonist by administering a polymer conjugate of the present invention.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2017513917-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2010521466-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2013151563-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2017513918-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2014532728-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2012502904-A
http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2010509227-A
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