http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2005504130-A
Outgoing Links
Predicate | Object |
---|---|
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J73-005 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J75-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J73-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07J7-00 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J75-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J73-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07J7-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B53-00 |
filingDate | 2002-09-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 2005-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | JP-2005504130-A |
titleOfInvention | Process for producing 17β- (substituted) -3-oxo-Δ1,2-4-azasteroids and intermediates |
abstract | OR 2 where R 1 is C 1 -C 4 alkyl and R 2 is a C 1 -C 4 alkyl radical, or R 3 and R 4 are equal or different, hydrogen or C 1 -C 4 alkyl to a radical, 17.beta. (substituted) -3-oxo - [delta 1, 2-4-aza-steroids (I) are 2- (substituted) of formula (IV) R 5 is Br or trichloromethyl sulfonyl -3 -It can be obtained by a method comprising the step of cleaving the oxazolidinedione ring present in hydroxyoxazolidinedione and removing the substituent at the 2-position to form a double bond at the 1,2-position. A part of compound (I) is a testosterone-5α-reductase inhibitor and can be used for the treatment of hyperandrogenic diseases. [Chemical 1] |
priorityDate | 2001-09-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 20.