http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2005035978-A
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_2cc87d476fde0ce82ac3b7245e61b785 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C221-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B61-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07B53-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D307-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D307-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C223-02 |
filingDate | 2004-05-24-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_80e0f01107459e8657e5d0192b579dec http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6f4299d1c5f1f7a22fa43beeb7edc5fe |
publicationDate | 2005-02-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | JP-2005035978-A |
titleOfInvention | Process for producing optically active form of syn-α-alkyl-β-aminocarbonyl compound |
abstract | The present invention provides a method for producing a corresponding syn-α-alkyl-β-aminocarbonyl compound with high yield, high syn selectivity, and high enantioselectivity. An aniline derivative (3) is reacted with an aldehyde (2) to give an imine (4), and the imine is reacted with an aldehyde (5) in the presence of a proline derivative (6). -Production method of optically active substance (1) of aminocarbonyl compound. [Chemical 1] [R 1 represents an aryl group, an aroyl group, a heterocyclic group or the like, R 2 , R 3 and R 4 represent a hydrogen atom, a halogen atom, an alkyl group or an alkoxy group, and R 5 represents a hydrogen atom, an alkyl group or Represents an alkenyl group, R 6 represents a hydrogen atom, an alkyl group or an alkenyl group, and A represents a hydrogen atom, an alkoxy group, an aryloxy group, an acyloxy group or a (substituted) silyloxy group. ] [Selection figure] None |
isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/WO-2008084750-A1 http://rdf.ncbi.nlm.nih.gov/pubchem/patent/CN-102584632-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2007182419-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2016108254-A http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2008169160-A |
priorityDate | 2003-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 136.