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filingDate 2001-06-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2004-03-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2004507232-A
titleOfInvention Methods for separating non-nuclear regulatory-mediated activity from steroid receptor-mediated nuclear transcription-regulating activity
abstract The present invention relates to a basic discovery in understanding the mechanism of action that is not mediated by steroid nuclear transcription control and its relationship to effects through steroid nuclear transcription control. (I) that effects that do not and do not through nuclear transcription control can be mediated by the same steroid receptor; (ii) both effects are induced by the ligand; (iii) rapid and That ligand-induced activation of the slowly adaptable ligand-binding domain exerts effects that are not through nuclear transcriptional regulation; (iv) steroids, which are typically the result of slower and stronger interactions Ligand-induced activation of the DNA binding domain of the receptor exerts an effect through nuclear transcriptional regulation; (v) the effect of ligand interaction without nuclear transcriptional regulation affects the selective response It has been discovered that ligand interactions can be related in this manner to effects through nuclear transcriptional regulation. The present invention also describes for the first time that certain steroids can induce effects that are not through nuclear transcriptional control through binding to an unrelated steroid receptor.
isCitedBy http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2007306885-A
priorityDate 2000-06-13-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID514876
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCO28185
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ72XC1
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID23426
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2S1C9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4VYI0
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP22498
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID18171
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ5XC70
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9JV42
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP59490
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9E6P5
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ9HVC3
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB5E572
http://rdf.ncbi.nlm.nih.gov/pubchem/taxonomy/TAXID11757
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ88Z39
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP21944
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID945041
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID15020
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB2S4P8
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ7V342
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID796
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ4UNV0
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID57976491
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0K466
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP07453

Total number of triples: 1938.