http://rdf.ncbi.nlm.nih.gov/pubchem/patent/JP-2003535061-A

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filingDate 2001-05-08-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2003-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2003535061-A
titleOfInvention Conjugates of endothelin receptor antagonists and antiepileptic compounds or analgesics with pain-relieving properties
abstract (57) [Summary]nThe present invention is independently selected from the group consisting of a pain-relieving effective amount of an endothelin antagonist or a pharmaceutically acceptable salt thereof, and an antiepileptic compound having analgesic properties and an analgesic and a pharmaceutically acceptable salt thereof. A new compound effective for reducing pain containing 1 to 3 kinds of compounds, and a pharmaceutical composition containing the same. The administration of endothelin receptor antagonists in these new conjugates can improve the frequency and severity of pain. The new conjugates described above can reduce the incidence of unwanted side effects as compared to higher doses of a single drug used to achieve the same therapeutic effect. The present invention also relates to new conjugates for the treatment of pain in mammals, including humans, and methods of using effective amounts of the pharmaceutical compositions thereof.
priorityDate 2000-05-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID5743
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID1775
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426106203
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424396562
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID10119029
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID282648
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422200240
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID69422924
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53240995
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424396569
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422200241
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID53241087
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID424396570
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422201451
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID4601
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422200252
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http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID57438043
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Total number of triples: 1024.