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filingDate 1999-01-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationDate 2002-03-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2002509120-A
titleOfInvention Pharmaceutical formulations and methods for their preparation
abstract (57) [Summary]nA pharmacologically effective amount of a pharmaceutical compound having amidine-based groups and optional ester groups, or a pharmaceutically acceptable salt thereof, a pharmaceutically acceptable solid carrier, and at the most stable pH A pharmaceutical composition comprising a tablet or capsule containing an amount of a pharmaceutically acceptable acid that substantially adjusts the pH of the composition to the pH of the compound. Such compositions are prepared by adding water during the manufacture of the formulation, and adding the compound to a pharmaceutically acceptable acid whose pH in a saturated aqueous solution is substantially the pH of the compound at the pH of highest stability. It is prepared by contact during the manufacture of the formulation.
priorityDate 1998-01-16-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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