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publicationDate 2002-11-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber JP-2002332297-A
titleOfInvention Bioactive compounds tyropeptins A and B and their production
abstract (57) [Problem] To provide a compound having a novel molecular skeleton exhibiting proteasome inhibitory activity. SOLUTION: The following formula (I) Tyropeptin A represented by the following formula (II) Is a novel proteasome inhibitor, Kitasatospora sp. Strain MK993-dF2 (FE RM P-18233). Tyropeptin A And tyropeptin B is a compound having proteasome inhibitory activity and useful as an antitumor agent.
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