abstract |
(57) [Summary] General formula (I): Wherein n is 0, 1 or 2; R 1 is hydrogen, alkyl, alkanoyl, cycloalkanoyl, (alkoxy) alkanoyl, aroyl, aryloxycarbonyl; R 2 is hydrogen, hydroxy, halo, alkoxy, alkanoyl Oxy, cycloalkanoyloxy, (alkoxy) alkanoyloxy, aroyloxy, aryloxycarbonyloxy; R 3 is pyrrolidinyl or piperidinyl] or a pharmaceutically acceptable salt thereof. Disclosed are methods of lowering plasma levels of La (a) or suppressing apo (a) production in humans by administering a sex vehicle. |