http://rdf.ncbi.nlm.nih.gov/pubchem/patent/IL-46683-A
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_3e9445e5e3626f36e932c6451a928250 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-044 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D495-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D495-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D491-044 |
| filingDate | 1975-02-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 1977-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | IL-46683-A |
| titleOfInvention | 2-alkyl-5-hydroxy-2,3-dihydro-1h-dibenzo(2,3:6,7)thiepino (oxepino) (4,5-c) pyrroles their production and pharmaceutical compositions containing them |
| abstract | 1499727 2,3 - Dihydro - 1H - debenzo- [2,3; 6,7]thiepino- or oxepino-[4,5-c]-pyrroles CIBA-GEIGY AG 13 Feb 1975 [22 Feb 1974] 6150/75 Heading C2C Novel compounds I and salts thereof in which X is O or S, R is OH or alkanoyloxy and R 1 is C 1-7 alkyl or C 1-7 alkenyl are prepared by (1) reacting a compound II in which X 1 and X 2 are reactive esterified hydroxy groups with an amine R 1 NH 2 or (2) alkylating or alkenylating a compound IV compounds I (R = OH) are also prepared by hydrolysing a corresponding ether or ester derivative or by diazotization of a 5-amino group; compounds I (R = alkanoyloxy) are also prepared by acylating a compound I (R = OH); and a compound I obtained may be converted into the salts or a salt thereof converted to the corresponding free base. Compounds I have CNS-depressant and agitation-inhibiting activity and form with a carrier a pharmaceutical composition which may be administered orally or parenterally.n[GB1499727A] |
| priorityDate | 1974-02-22-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 98.