http://rdf.ncbi.nlm.nih.gov/pubchem/patent/HU-T78121-A
Outgoing Links
| Predicate | Object |
|---|---|
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-365 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D491-052 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D495-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-47 |
| filingDate | 1995-12-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2ca9f6692da47b7e7939bafde8515a8f http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_678c9d1db82afaffe7b963c54bf991d4 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9d89619b35d0e87f4db43e8210beaf8b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b9f88406f8aa69775b599c17f5b3841e http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_122c4d68eb54a1628feab4b6644eaae5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_42811bdfc4f7bfb002baf61349fef9cc http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_84d3aac72adaa189e61557aeef8925f0 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8844ac1c7c9c7939e2c44f6e63c7a3fe http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3dd83b06f2be608dc0014245cc907c06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_09af6cda955badcb1ccddc1a20f4ad30 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2b708ae6ae283073cbba40564859bffb |
| publicationDate | 1999-12-28-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | HU-T78121-A |
| titleOfInvention | Androgen receptor modulator condensed quinoline and indole derivatives, process for their preparation, use and pharmaceutical compositions containing them |
| abstract | Cpds. of formula e.g. (I), (II), (VII) and (XII) are new: (I) = (A; X1 = R1); (II) = (A; X1 = a gp. of formula (i)); (VII) = (C; either K = CR3 and L = CH or K = CHR3 and L = CH2); (XII) = (C; K = CR3R21 and L = C=X); R1 = heteroaryl opt. substd. by 1-4C alkyl, F, Cl, Br, NO2, CO2H, CO2R2, CHO, CN, CF3, CH2OH or COMe, and is attached through C or N atom; R2 = H, 1-4C alkyl or perfluoroalkyl, aryl, heteroaryl or opt. substd. allyl, arylmethyl, alkynyl or alkenyl; R3 = H, 1-4C alkyl or perfluoroalkyl, hydroxymethyl, aryl, heteroaryl or opt. substd. allyl, arylmethyl, alkynyl or alkenyl; R4-R6, R11-R15 = H, F, Cl, Br, I, NO2, CO2H, CO2R2, CN, CF3, CH2OH, 1-4C alkyl or perfluoroalkyl, OR2, SR2, S(O)R2, SO2R2, SO3H, S(NR2R7)R2, S(O)(NR2R7)R2, NR2R7, aryl, heteroaryl or opt. substd. allyl, arylmethyl, alkynyl or alkenyl; R7 = H, 1-4C alkyl or perfluoroalkyl, aryl, heteroaryl, opt. substd. allyl or arylmethyl, OR8 or NHR8; R8 = H, 1-6C alkyl or perfluoroalkyl, aryl, heteroaryl, opt. substd. allyl or arylmethyl, SO2R2 or S(O)R2; R9, R10 = H, 1-6C alkyl or perfluoroalkyl, aryl, heteroaryl or opt. substd. allyl, arylmethyl, alkynyl or alkenyl; or R9 + R10 = 3-7 membered ring opt. substd. by H, F, OR2 or NR2R7; X = CH2, O, S or NR7; R20 = 1-6C alkyl or opt. substd. allyl, arylmethyl, alkenyl, aryl or heteroaryl; R21 = H, 1-4C alkyl or opt. substd. allyl, arylmethyl, aryl or heteroaryl; with provisos. |
| priorityDate | 1995-12-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 447.