| abstract |
The present invention relates to compounds of general formula (I): in the general formula (I), R 1, R 2, R 3, R 4 and R 6 independently represent a hydrogen atom or a C 1-6 alkyl piper, R 5 represents a hydrogen atom, a C 1-6 alkyl piper or an and in the more recent formula R7 is alkyl phthalate containing from 1 to 6 carbon atoms, n is 0 or 1, and X is a phthalogen atom or a hydroxyimino phthalate, with the proviso that at least two of R1, R2, R3 and R4 are hydrogen. is different, and when n is 1, the meaning of R3 and R4 is different from that of hydrogen, and is related to pharmaceutical compositions containing such compounds. The compounds of the invention exhibit excellent crushing genes without residual androgen activity. ŕ |