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filingDate 2001-03-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f46a2bbb32ee9e8d615057e7d4aa02d2
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_200490a3345d8b0232c265b593b85566
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http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51b671ab428c2f3eb75c9857a818c3e4
publicationDate 2013-11-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber HU-229348-B1
titleOfInvention A process for the preparation of epothilone analogs and intermediates
abstract The present invention relates to a process for the preparation of epothilone analogs by initially forming novel ring-opended epothilones and carrying out a macrolactamization reaction thereon. The subject process is amenable to being carried out in a single reaction vessel without isolation of the intermediate compound and provides at least about a threefold increase in yield over prior processes for preparing the desired epothilone analogs.
priorityDate 2000-03-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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