http://rdf.ncbi.nlm.nih.gov/pubchem/patent/HR-P20120627-T1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_12a9e9ce63eb0bbf3658453fb50a6d9b |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-08 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-4866 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H23-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H15-26 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-2018 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K9-0019 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H15-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07H15-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P39-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-351 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-70 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P3-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-7004 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H15-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H15-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07H15-26 |
| filingDate | 2012-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_87a21ed2cbc2deb90f400577eed11195 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_dc013f168052db85855ea1fb7ce224d3 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_6711592674231243013757cefdbb75b6 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_e58a6469f5a82ed4e16e7e3166243e37 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eac22a42529c3f98baa2d941cef258e6 |
| publicationDate | 2012-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | HR-P20120627-T1 |
| titleOfInvention | GLUCOPIRANOSIL-SUBSTITUTED BENZOL DERIVATIVES, THE MEDICINAL PRODUCTS CONTAINING THESE COMPOUNDS, THEIR USE AND THE PROCESS OF THEIR PRODUCTION |
| abstract | Glucopyranosyl-substituted benzene derivatives having the general formula I wherein R 1 is selected from the following meanings: hydrogen, fluorine, chlorine, bromine, iodine, C 1-4 alkyl, C 2-6 alkynyl, C 1-4 alkoxy, C2-4-alkenyl-C1-4-alkoxy, C2-4-alkynyl-C1-4-alkoxy, methyl substituted by 1 to 3 fluorine atoms, ethyl substituted by 1 to 5 fluorine atoms, methoxy substituted by 1 to 3 fluorine atoms , ethoxy substituted with 1 to 5 fluorine atoms, C1-4-alkyl substituted by a hydroxy- or C1-3-alkoxy group, C2-4-alkoxy substituted by a hydroxy- or C1-3-alkoxy group, C2-6- alkenyl, C3-6-cycloalkyl, C3-6-cycloalkyl-C1-3-alkyl, C3-7-cycloalkyloxy, C3-6-cycloalkyl-C1-3-alkoxy, C5-7-cycloalkenyloxy, hydroxy, amino, nitro or cyano, while in the C5-6 cycloalkyl groups the methylene group may be replaced by O, R2 denotes hydrogen, fluorine, chlorine, bromine, hydroxy, C1-4 alkyl, C1-4 alkoxy, cyano or nitro, while alkyl - or the alkoxy group may be mono- or poly-substituted with fluorine, and R3 is selected from the following z uses: tri- (C1-4-alkyl) silyl-C1-6-alkyl, C2-6-alkyn-1-yl, C2-6-alken-1-yl, amino, C1-3-alkylamino, di- ( C1-3-alkyl) amino, pyrrolidin-1-yl, pyrrolidin-2-one-1-yl, piperidin-1-yl, piperidin-2-one-1-yl, morpholin-4-yl, morpholin-3- on-4-yl, piperazin-1-yl, 4- (C1-3-alkyl) piperazin-1-yl, nitro, C3-7-cycloalkyloxy, C5-7-cycloalkenyloxy, C3-7-cycloalkylsulfanyl, C3-7 -cycloalkylsulfinyl, C3-7-cycloalkylsulfonyl, C5-7-cycloalkenylsulfanyl, C5-7-cycloalkenylsulfinyl and C5-7-cycloalkenylsulfonyl, while the above alkynyl- and alkenyl groups may be mono- or poly-substituted with fluorine or chlorine, preferably with fluorine, and wherein the above alkynyl and alkenyl groups may be mono- or di-substituted with the same or different L1 groups; wherein said cycloalkyl and cycloalkenyl rings may independently of one another be mono- or di-substituted by substituents selected from fluorine and C1-3-alkyl, and while in the above-mentioned cycloalkyl and cycloalkenyl rings, one or two methylene groups may be substituted independently of one another with O, S, CO, SO, SO2 or NRN, preferably with O, CO, S, SO2 or NRN, preferably with O or CO, R4, R5 independently of one another denote hydrogen, fluorine, chlorine, bromine, iodine, cyano, nitro , C1-3-alkyl, C1-3-alkoxy, methyl or methoxy substituted by 1 to 3 fluorine atoms, RN denotes H, C1-4-alkyl, C1-4-alkylcarbonyl or C1-4-alkylsulfonyl, L1 are independently selected from hydroxy-, cyano-, nitro-, C3-7-cycloalkyl-, aryl-, heteroaryl-, C1-4-alkylcarbonyl-, arylcarbonyl-, heteroarylcarbonyl-, aminocarbonyl-, C1-4-alkylaminocarbonyl-, di - (C1-3-alkyl) aminocarbonyl-, pyrrolidin-1-ylcarbonyl-, piperidin-1-ylcarbonyl-, morpholin-4-ylcarbonyl, arylaminocarbonyl-, heteroarylaminocarbonyl-, C1-4-alkoxy icarbonyl-, aryl-C1-3-alkoxycarbonyl-, heteroaryl-C1-3-alkoxycarbonyl-, C1-4-alkyloxy-, aryloxy-, heteroaryloxy-, C1-4-alkylsulfanyl-, arylsulfanyl-, heteroarylsulfanyl-, C1-4 -alkylsulfinyl-, arylsulfinyl-, heteroarylsulfinyl-, C1-4-alkylsulfonyl-, arylsulfonyl- |
| priorityDate | 2004-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 77.