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publicationDate 2020-11-11-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber GB-2583882-A
titleOfInvention Compounds
abstract Compounds of general formula (I): wherein R1, R2, R3, R4, R5a, R5b X1, X2, Z and Y are as defined herein are positive modulators of the calcium-activated chloride channel (CaCC), TMEM16A. The compounds are useful for treating diseases and conditions affected by modulation of TMEM16A, particularly respiratory diseases and conditions.
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Total number of triples: 665.