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filingDate 2012-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9f1153d332f9ef7c3ad30d09d34dcb4c
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publicationDate 2013-08-28-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber GB-2499666-A
titleOfInvention Mcl-1 inhibitors for the treatment of conditions associated with proliferative disorders
abstract The invention relates to use of compounds represented by the general formula (I) : and pharmaceutically acceptable salts thereof, wherein n is an integer from 2 to 5; p is an integer from 0 to 4; R1 is independently selected from the group consisting of a hydroxl group, an alkoxy group, a thiol group, and a thioether group, wherein at least two of R1 are on the carbon-2 and carbon-5 positions of the phenyl group; R2 and R3 are independently a methylene group or a nucleophile; Z is an oxygen (O) atom or sulfur (S) atom; and T is hydrogen or an optionally substituted aliphatic group or optionally substituted aryl group; in the manufacture of a medicament for prevention and/or treatment and/or containment of a condition associated with a cell proliferative disorder. Particular conditions include tumorigenesis and cancer.
priorityDate 2012-02-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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