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filingDate 2009-03-31-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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publicationDate 2010-01-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber GB-2462022-A
titleOfInvention Controlled release compositions for use in reducing circulating levels of platelets
abstract Use of a controlled release composition comprising a platelet reducing agent having a 3 month shelf stability for use in the treatment and/or prevention of platelet related conditions or disorders including haematological proliferative disorders, myloproliferative disorders and thrombotic and vaso-occulsive disorders. The composition may comprise a solid support core; an optional preparatory coat; a substrate layer comprising a binder and microparticles of a platelet number reducing agent such as anagrelide or a derivative thereof which is present in a form that has a shelf stability of at least 3 months; a release control component effective for the controlled release of the platelet number reducing agent; and an optional finishing coat and/or enteric coating. The composition may further comprise a seal coat layer which may be dispersed between the substrate layer and the release control component. The composition may be administered together with other therapeutic agents. Methods and pharmaceutical preparations comprising such agents are also provided.
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Total number of triples: 1463.