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publicationDate 1994-04-20-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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titleOfInvention HIV integrase inhibitors
abstract Compounds of the general formula: <IMAGE> wherein n is 0-3; p is 1-2; q is 1-2; X is CH2, O or N-R<1>, and R<1> is H, C1-4alkyl or C3-5cycloalkyl; R is (a) C1-6 alkyl; (b) C1-6alkoxy; (c) hydroxyl; (d) halogen; (e) CN; (f) NO2; (g) NHSO2CHÏ; or (h) COOH; G is H or R, and salts or hydrates thereof have HIV integrase inhibiting activity.
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