http://rdf.ncbi.nlm.nih.gov/pubchem/patent/GB-1469679-A
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_bee8b2c674d7ec672688001f27aa95fe |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D223-20 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D223-20 |
| filingDate | 1974-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 1977-04-06-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | GB-1469679-A |
| titleOfInvention | 1-amino-5,6-dihydro-morphanthridine-5,11-dione compounds and processes for their preparation |
| abstract | 1469679 1 - Amino - 5,6 - dihydromorphanthridine - 5,11 - dione derivatives CHEM PHARMAZ FABRIK DR HERMANN THIEMANN GmbH 10 Dec 1974 [10 Dec 1973] 53324/74 Heading C2C Novel compounds of Formula I wherein R 1 and R 2 , which may be the same or different, each represents a hydrogen or halogen atom or a methyl, methoxy, methylthio, trifluoromethyl, nitro or acetyl radical, wherein at least one of the radicals represented by R 1 and R 2 is a hydrogen atom, R 3 represents a lower alkyl radical or a hydrogen atom, R 4 represents a lower alkyl radical or the radical in which n represents 0 or an integer from 1 to 3, and Y represents a halogen atom or an amino, mono - (lower - alkyl) - amino, di - (loweralkyl) - amino, piperidino, piperazino, or morpholino radical, and R 5 represents a hydrogen atom or a lower alkyl radical and lower denotes groups containing 1 to 3 carbon atoms, are prepared either (a) from a compound of Formula II which is mono- or di-alkylated at the 1-amino group or reacted with an #-haloalkanoic acid halide or phosgene and then with HY or (b) reacting a compound of Formula III wherein R 6 is C 1-3 alkyl with hydrazoic acid. Pharmaceutical compositions in conventional forms for oral, rectal and parenteral administration and having tranquillizing, neuroleptic and cramp relieving activity comprise an above novel compound and a carrier or diluent. |
| isCitedBy | http://rdf.ncbi.nlm.nih.gov/pubchem/patent/EP-0089322-A1 |
| priorityDate | 1973-12-10-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 23.