http://rdf.ncbi.nlm.nih.gov/pubchem/patent/FR-2842735-A1

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filingDate 2002-07-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_eb2c7ee773ba75ba32ab5a03ba07b6ef
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3cd163f1716235b9fd4752560017bead
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publicationDate 2004-01-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber FR-2842735-A1
titleOfInvention MODIFIED RELEASE MICROCAPSULES OF LOW SOLUBLE ACTIVE PRINCIPLES FOR PER OS ADMINISTRATION
abstract The present invention relates to microcapsules allowing the modified release in a reliable and industrially reproducible manner of a principle (AP) which is poorly soluble in water, to the exclusion of antihyperglycemic agents. Each of these microcapsules comprises a core of poorly soluble AP and a coating film applied to the core. Their average diameter is less than 1000 microns. The coating film contains a film-forming polymer (P1) insoluble in the fluids of the gastrointestinal tract; a water-soluble polymer (P2); a plasticizer (PL); and optionally a lubricating surfactant (TA). This coating film represents at least 4% w / w dry of their total mass, and its components P1, P2, PL satisfy the following characteristics: mass fraction by dry weight of P1 relative to the total mass of the coating, between 40 and 90%; mass fraction by dry weight P2 / P1 + P2 between 15 and 60%; mass fraction by dry weight PL / P1 + PL between 1 and 30%. The invention also relates to the applications of said microcapsules in galenics.
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priorityDate 2002-07-26-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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