http://rdf.ncbi.nlm.nih.gov/pubchem/patent/FI-114153-B
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_d225eacc0d6d94f83eeeaaba9abc4f21 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D231-44 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N- http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D- |
| filingDate | 1995-04-18-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2004-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_155a92a75dff99a41a1e21e5ea245902 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c9fdffab5727855346840e9667125b8f http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a7b7104da4c4713955cbb21d95b19065 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_829851925146fb2321691d6156a2dd69 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_47711c646ad5101969ee419592a0dc16 |
| publicationDate | 2004-08-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | FI-114153-B |
| titleOfInvention | Process for preparation of N-phenylpyrazole derivatives having therapeutic effect |
| abstract | N-phenylpyrazole derivs. of formula (I) are new: where R1 = CN, NO2, halo, Ac or CHO; R2 = R5SO2, R5SO or R5S; (R5 = opt. branched alkyl, alkenyl or alkynyl of up to 4C, opt. substd. by opt. different halogen(s)); R3 = H, halo, -NR6R7, opt. branched alkoxymethyleneamino contg. 2-5C and opt. substd. on the CH2 by an opt. branched 1-4C alkyl gp. or opt. branched 2-5C alkoxycarbonyl opt. substd. by halogen(s); (R6, R7 = H, opt. branched alkyl, alkenylalkyl, or alkynylalkyl of up to 5C, CHO or 2-5C opt. branched alkanoyl or haloalkanoyl; or NR6R7 = 5-or 6-membered cyclic imide); R4 = phenyl substd. in the 2-posn. by F, Cl, Br or I; in the 4-posn. by opt. branched 1-4C alkyl or alkoxy (opt. substd. by halogen(s)) or a Cl or Br; and opt. in the 6-posn. by F, Cl, Br or I; with the exclusion of the cpd. where R1 = Cn, R2 = MeSO2, R3 = NH2 and R4 = 2,6-dichloro-4-tri fluoromethylphenyl. Pref. in (I): (i) R1 is not CHO and neither R6 or R7 is alkenylalkyl or alkynylalkyl; (ii) R2 = 1-4C alkylsulphonyl/sulphinyl/thio opt. halogen substd. or up to 4C alkenyl- or alkynyl-sulphonyl/sulphinyl/thio opt. halogen substd.; R3 = H, NH2, or NHMe; and R1 = halogen, or esp. CN or NO2; and esp. (iii) R4 contains a CF3 or OCF3 gp.; and R2 = opt. halogenated 1-4C alkylsulphionyl/sulphinyl/thio gp.; partic. R2 = SCF3, SOCF3, or SO2CF3; and R4 = 2,4,6-trichloro-, or 2,6-dichloro-4-difluoromethoxy-, 2-chloro-4-trifluoromethyl-,etc. |
| priorityDate | 1987-06-12-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 475.