http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-420179-A1
Outgoing Links
Predicate | Object |
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assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_966a6c1f382ec9bcb5e3839dfd73e5b8 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D337-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07C65-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D313-12 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D313-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C251-50 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C249-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D337-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C65-36 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07C251-20 |
filingDate | 1973-11-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 1976-05-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | ES-420179-A1 |
titleOfInvention | A PROCEDURE FOR THE PREPARATION OF TRICYCLIC IMINES WITH PHARMACODYNAMIC ACTIVITY. |
abstract | A procedure for the preparation of tricyclic imines, with pharmacodynamic activity, of the general formula ** (See formula) ** wherein X represents a sulfur atom, an oxamethylenic or thiamethylene group, an ethylenic group (which may be substituted by lower alkanoylamide) or a vinyllenic group (which may be substituted by halogen, lower alkyl, cyano or sulfamoyl) ; R1 represents a hydrogen or halogen atom or a group of hydroxyl, lower alkoxy, lower alkyl, cyano, lower alkoxycarbonyl, carbamoyl, sulfamoyl, lower alkyl mercapto, trifluoromethyl or nitro; R2 and R3 individually represent a hydrogen atom or a lower alkyl group, or both, together with the nitrogen atom to which they are attached, represent a saturated, pentagonal or hexagonal monocyclic heterocyclic group, which may contain an oxygen atom or sulfur or one more nitrogen atom; R4 represents a hydrogen atom or a lower alkyl group; m represents an integer valued from 1 to 3; and n represents an integer valued from 2 to 5, and its acid addition salts, characterized in that a compound of the general formula is reacted ** (See formula) ** wherein X, R1, R4, m and n have the same meaning as indicated above, while Y represents a halogen atom, a lower alkylsulfonyloxy group or a phenylsulfonyloxy group (which may be substituted by lower alkyl or halogen), with an amine of the general formula ** (See formula) ** where R2 and R3 have the same meaning as before, and if desired, converting a compound of formula I to an acid addition salt. (Machine-translation by Google Translate, not legally binding) |
priorityDate | 1970-10-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 28.