http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-393757-A1
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_fdaa64756184e715af6cb25ebc318917 |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D205-09 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D205-095 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D205-095 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D205-09 |
filingDate | 1971-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationDate | 1975-09-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | ES-393757-A1 |
titleOfInvention | A METHOD FOR THE PREPARATION OF AZETIDIN-2-ONAS. |
abstract | A method for the preparation of azetidin-2-ones containing a thio-substituent at position 4 of the ring, of formula: ** (See formula) ** where X is halogen, an azido group or an imido group derived from a dicarboxylic acid; R is an alkyl or aralkyl group; R1 is an alkoxy or aralkoxy group; R2 and R3 are the same or different and each represents hydrogen, alkyl, aralkoxy or alkylthioalkyl; Y and Z are both hydrogen and when taken together represent a bond between the carbon atoms to which they are attached, the method of which is to react a thioimidate derivative of an α-amino acid ester with a monosubstituted acetyl halide of the formula I: X.CH.CO.Hal (I) where X is halogen, an azido group or an imido group derived from a dicarboxylic acid and the symbol -Hal- represents halogen, under anhydrous conditions and in the presence of a tertiary base. (Machine-translation by Google Translate, not legally binding) |
priorityDate | 1970-07-31-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 20.