http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-349316-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_2e5edd48190cba3fa70dd3975efd9831 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-86 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-70 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D277-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-485 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-74 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-445 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/E02F9-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D211-90 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-86 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K- http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-90 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/E02F9-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-445 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-74 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D211-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-485 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D277-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-04 |
| filingDate | 1968-01-15-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 1969-04-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-349316-A1 |
| titleOfInvention | PROCEDURE FOR THE PREPARATION OF 4,5,6,7-TETRAHYDRO - THIAZOLO (5,4-C) PYRIDINES. |
| abstract | Novel compounds of the formula (wherein R 1 is H, C 1-6 alkyl, C 2-6 alkenyl, halo C 2-6 alkenyl, C 3-8 cycloalkyl, C 6-10 aryl, C 7-9 aralkyl, aromatic or aliphatic carboxylic or sulphonic acyl, carbamoyl or amidino R 2 is H, C 1-6 alkyl, C 2-6 alkenyl, halo C 2-6 alkenyl, or cycloalkyl, or NR 1 R 2 is a heterocyclic ring which may contain a further hetero atom and/or be OH, methyl or phenyl substituted R 3 is H, C 1-6 alkyl, C 2-6 alkenyl, halo C 2-6 alkenyl, C 3-8 cycloalkyl, C 6-10 aryl, C 7-9 aralkyl, aromatic or aliphatic carboxylic or sulphonic acyl, carbamoyl, thiocarbamoyl or amidino and where alkyl groups R 1 , R 2 and/or R 3 may be OH, alkoxy, aryloxy, cycloalkyl, carboxy, carbalkoxy or amido substituted, and aromatic groups R 1 , R 2 and/or R 3 may be halogen, OH, alkyl, alkoxy, alkylthio, alkylsulphonyl, alkylenedioxy, amino, alkylamino, acylamino or aminosulphonyl substituted. R 4 and R 5 are H, alkyl, aryl or aralkyl and R is a bond or a C 1-3 hydrocarbon chain) and acid-addition salts thereof, are prepared from hydrohalic acid salts of the appropriate 3-bromo-4-piperidones and thioureas or thioamides. Products wherein R 3 is aryl may be hydrolysed, provided R 1 is not aryl, to the corresponding compounds wherein R 3 is H, which compounds may in turn be reacted with appropriate reagents to replace the H atom R 3 by another radical or group R 3 (except aryl). |
| priorityDate | 1965-07-23-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 41.