http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-335760-A1
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_14effe3850d2129f863b969dac4f1db8 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D295-13 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D281-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D295-195 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D267-20 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D295-195 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D295-13 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D267-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D281-16 |
| filingDate | 1967-01-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationDate | 1968-03-16-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-335760-A1 |
| titleOfInvention | PROCEDURE FOR THE PREPARATION OF TIAZE-PINE DERIVATIVES. |
| abstract | Process for the preparation of thiazepine derivatives of general formula ** (See formula) ** wherein R means lower alkyl, R1 and R2 mean hydrogen, lower alkyl, lower alkoxy, halogen, nitro or trifluoromethyl, Y means hydroxyl, amino, lower alkylamino, lower dialkylamino, lower alkoxy, 1-piperazino, 4- (lower alkyl ) -1-piperazino, 4- (hydroxy-lower alkyl) -1-piperazino, pyrrolidino, lower alkyl pyrrolidino, piperidino, lower alkyl piperidino, morpholino or lower alkyl morpholino and the group (see formula) and the radical as a whole, represents 1-piperazino, 4- (lower alkyl) -1-piperazino or 4- (hydroxy-lower alkyl) -1-piperazino, in which R and Y have the above definition and n is an integer from 2 to 4, characterized in that it comprises: cyclizing a compound of general formula ** (See formula) ** where E means (see formula) or a convertible group in it, and B, ne Y have the definition above, R1 and R2 have the definition above or mean transformable radicals in it, F or C mean mercapto and the other is halogen, nitro or thiazonium and in which F and G can occupy exchanged positions, to form a heterocyclic ring in which F and G together form the -S-; convert if necessary, before or after said cyclization, E in the group (see formula) and if necessary, before or after said cyclization, when one of R1 or R2 is amino, it is transformed into hydrogen, lower alkoxy or halogen. (Machine-translation by Google Translate, not legally binding) |
| priorityDate | 1966-01-17-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 24.