abstract |
A compound selected from the group consisting of: N- (4- (4- (2- (tert-butyl) -6-methylpyrimidin-4-yl) piperazin-1-yl) butyl) -4-phenylpiperazine-1-carboxamide , N- (4- (4- (6- (tert-butyl) -2-methylpyrimidin-4-yl) piperazin-1-yl) butyl) -4-phenylpiperazine-1-carboxamide, N- (4- (4 - (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4-yl) piperazin-1-yl) butyl) -4-phenylpiperazine-1-carboxamide, 4-phenyl-N- (4- (4- (quinolin-4-yl) piperazin-1-yl) butyl) piperazine-1-carboxamide, N- (4- (4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4-yl) piperazin -1-yl) butyl) -3- (pyridin-4-yl) azetidine-1-carboxamide, N- (4- (4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4-yl ) piperazin-1-yl) butyl) -5-methoxyisoindoline-2-carboxamide, N- (4- (4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4-yl) piperazin-1- yl) butyl) -4,5-dihydro-1H-benzo [d] azepine3 (2H) -carboxamide, N- (4- (4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4- il) piperazin-1-yl) butyl) -4-phenylpiperidine-1-carboxamide, N- (4- (4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4-yl) piperazin-1 -il) butyl) -3 , 4-dihydro-1H-pyrido [4,3 -b] indole-2 (5H) -carboxamide, N- (4- (4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4- yl) piperazin-1-yl) butyl) -4-phenylcyclohexanecarboxamide, 4-phenyl-N- (4- (4- (quinolin-4-yl) piperazin-1-yl) butyl) cyclohexanecarboxamide, N- (4- ( 4- (2- (tert-butyl) -6- (trifluoromethyl) pyrimidin-4-yl) piperazin-1-yl) butyl) imidazo [1,2-a] pyridin-2-carboxamide, and / or a pharmaceutically acceptable salt acceptable thereof. |