http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2692720-T3

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filingDate 2014-07-29-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5612731d3eb320da9a7df7d791b42d4f
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f1bdaff5fa508d0a990f3273564516f2
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cf2182fdda0927feb17c1c87d5cddf09
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publicationDate 2018-12-04-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2692720-T3
titleOfInvention 1,2-disubstituted cyclobutyl compounds
abstract A compound of the general Formula (I), or a pharmaceutically acceptable salt, a stereoisomer, an amide, an ester, a carbamate, a carbonate, a ureido, a phosphate or a biohydrolizable solvate thereof: ** Formula ** in that R1 is selected from the group consisting of substituted or unsubstituted aryl and substituted or unsubstituted heteroaryl; R 2 and R 3, identical or different, are selected from the group consisting of hydrogen, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted cycloalkylalkyl and substituted or unsubstituted alkenyl; or R2 and R3 together with the bridge nitrogen atom to which a substituted or unsubstituted non-aromatic heterocyclyl are attached, in which the aryl, heteroaryl or heterocyclyl groups can be substituted, independently, in one or more available positions, with one or more suitable groups selected from OR ',> = O, SR', SOR ', SO2R', OSO2R ', OSO3R', NO2, NHR ', N (R') 2,> = N-R ', N (R ') COR', N (COR ') 2, N (R') SO2R ', N (R') C (> = NR ') N (R') R ', N3, CN, halogen, COR', COOR ', OCOR', OCOOR ', OCONHR', OCON (R ') 2, CONHR', WITH (R ') 2, PO (OR') 2, PO (OR ') R', C1-C12 alkyl, C3 cycloalkyl -C10, C2-C12 alkenyl, C2-C12 alkynyl, aryl, heteroaryl and non-aromatic heterocyclic group, in which each of the R 'groups is independently selected from the group consisting of hydrogen, OH, NH2, SH, CN, halogen, COH, CO-alkyl, COOH, C1-C12 alkyl, C3-C10 cycloalkyl, C2-C12 alkenyl, C2-C12 alkynyl, aryl, heteroaryl and non-aromatic heterocyclic group.
priorityDate 2013-07-30-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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