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filingDate 2014-03-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2018-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b36f16333d2aaa2eb5496844de8b90a3
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_140fb8981838b5e55e93bbf7288c4bbc
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publicationDate 2018-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2689526-T3
titleOfInvention P2X7 modulators
abstract A compound of Formula I ** Formula ** wherein: each R2 is independently selected from the group consisting of H, halo, SO2CH3, C1-C3 alkyl, NO2, NH2, perhaloalkyl and perhaloalkoxy; or two R2 substituents are taken together to form: ** Formula ** n is 0-3; X is H or C1-C3 alkyl; Y is independently selected from the group consisting of H, C1-C3 alkyl, and C3-C4 cycloalkyl; R1 is independently selected from the group consisting of: ** Formula ** Ra, Rc and Rg are independently H or halo; Rd is H or C1-C3 alkoxy; Re is independently selected from the group consisting of H, C1-C3 alkyl, and halo; Rb, Rf, Rh, Ri, Rj, Rk, Rl, Rm, Rn, Ro are independently selected from the group consisting of H, C1-C3 alkyl and perhaloalkyl; and Rp is H or C (O) OtBu; or a pharmaceutically acceptable salt of a compound of Formula (I).
priorityDate 2013-03-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 483.