http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2669793-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_40765ca9a78b54a8a76f781d159ad145 |
| classificationCPCAdditional | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-20 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D417-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-227 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-052 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D215-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P31-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D519-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-48 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-227 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D491-052 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D417-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-37 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D413-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D215-38 |
| filingDate | 2011-07-01-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2018-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_fc0dfc2f50db205d8b550aa18424e8dc http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b900db10f854af326e9f80fcd8c38844 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_cb63bdf3139fdf4c5e3dc1610631cdc7 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1aec92f4ec95e367cfd8d45b9a39f743 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_edfdecc2ce0b86d283118840abf71b6f http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_57a69defeb3fc7cafff080b748267566 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_399a8d8d7abd87c96ca0cf2e3b053071 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_03afd7d3054627ba07a9cd1b5cea4423 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_314786c4a77c4e9cba6c0960263e7a2b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_61e9466e0b55a8bde6299fc67ee2bf25 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_098c25bee7f4e1447eaa70f7133245d8 |
| publicationDate | 2018-05-29-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2669793-T3 |
| titleOfInvention | 2-quinolinyl-acetic acid derivatives as HIV antiviral compounds |
| abstract | A Compound of formula Ih: where: R1 is R1a or R1b; R4 is R4a or R4b; R5 is R5a or R5b; R6 is R6a or R6b; R7 is R7a or R7b; R1a is selected from: a) H, halo, (C1-C6) alkyl and (C1-C6) haloalkyl; b) (C2-C6) alkenyl, (C2-C6) alkynyl, (C3-C7) cycloalkyl, nitro, cyano, aryl, heterocycle and heteroaryl; c) -C (> = O) -R11, -C (> = O) -OR11, -OR11, -SR11, -S (O) -R11, -SO2-R11, - (C1-C6) alkyl-R11 , - (C1-C6) C (> = O) alkyl - R11, - (C1-C6) C-alkyl (> = O) -OR11, - (C1-C6) alkyl-OR11, - (C1-C6) alkyl-SR11, - (C1-C6) alkyl-S (O) -R11 and - (C1-C6) alkyl-SO2-R11, where each R11 is independently selected from H, (C1-C6) alkyl, (C2 -C6) alkenyl, (C2-C6) alkynyl, (C1-C6) haloalkyl, (C3-C7) cycloalkyl, aryl, heterocycle and heteroaryl; and d) -N (R9) R10, -C (> = O) -N (R9) R10, -OC (> = O) -N (R9) R10, -SO2-N (R9) R10, - (C1- C6) alkyl-N (R9) R10, - (C1-C6) alkyl- C (> = O) -N (R9) R10, - (C1-C6) alkyl-OC (> = O) -N (R9) R10 and - (C1-C6) alkyl-SO2-N (R9) R10, wherein each R9 is independently selected from H, (C1-C6) alkyl and (C3-C7) cycloalkyl, and each R10 is independently selected from R11 , - (C1-C6) alkyl-R11, -SO2-R11, - C (> = O) -R11, -C (> = O) OR11 and -C (> = O) N (R9) R11, where each R11 is independently selected from H, (C1-C6 alkyl), (C2-C6) alkenyl, (C2-C6) alkynyl, (C1-C6) haloalkyl, (C3-C7) cycloalkyl, aryl, heterocycle and heteroaryl; and wherein any aryl, heterocycle or heteroaryl of R1a is optionally substituted with one or more Z10 groups; R1b is selected from: a) - (C1-C6) alkyl-O- (C1-C6) alkyl- (C3-C7) carbocycle, - (C1-C6) alkyl-S- (C1-C6) alkyl- (C3 -C7) carbocycle, - (C1-C6) alkyl-S (O) - (C1-C6) alkyl- (C3-C7) carbocycle, - (C1-C6) alkyl-SO2- (C1-C6) alkyl- ( C3-C7) carbocycle, - (C1-C6) alkyl-SO2- (C1-C6) alkyl-Z13, - C (O) - (C1-C6) alkyl-Z13, -O- (C1-C6) alkyl- Z13, -S- (C1-C6) alkyl- Z13, -S (O) - (C1-C6) alkyl-Z13, -SO2- (C1-C6) alkyl-Z13, - (C1-C6) alkyl-Z14 , - (C1-C6) alkyl-C (O) - (C1-C6) alkyl-Z13, - (C1-C6) alkyl-C (O) -O (C1-C6) alkyl-Z13, - (C1- C6) alkyl-O- (C1-C6) alkyl-Z13, - (C1-C6) alkyl-S- (C1-C6) alkyl-Z13, - (C2-C6) alkenyl- (C1-C6) haloalkyl, - (C2-C6) alkynyl- (C1-C6) haloalkyl, - (C3-C7) halocarbocycle, -NRaSO2NRcRd, -NRaSO2O (C3-C7) carbocycle, -NRaSO2Oaryl, - (C2-C6) alkenyl- (C3-C7) carbocycle, - (C2-C6) alkenyl-aryl, - (C2-C6) alkenyl-heteroaryl, - (C2-C6) alkenyl-heterocycle, - (C2-C6) alkynyl- (C3-C7) carbocycle, - (C2 -C6) alkynyl-aryl, - (C2-C6) alkynyl-heteroaryl - (C2-C6) alkynyl-heterocycle, - (C3-C7) carbocycle-Z1 and -halo (C1-C6) alkyl-Z3, wherein any (C1-C6) alkyl, (C1-C6) haloalkyl, (C3 -C7) carbocycle, (C3-C7) halocarbocycle, (C2-C6) alkenyl, (C2-C6) alkynyl, aryl, heterocycle and heteroaryl, either alone or as part of a group, is optionally substituted with one or more Z1 groups; b) spiro-bicyclic carbocycle, fused bicyclic carbocycle and bridged bicyclic carbocycle, wherein any spiro-bicyclic carbocycle, fused bicyclic carbocycle and bridged bicyclic carbocycle is optionally substituted with one or more Z1 groups, where two Z1 groups together with the atom or atoms to which they are attached optionally form a (C3-C7) carbocycle or heterocycle, wherein the (C3-C7) carbocycle or heterocycle is optionally substituted with one or more Z1 groups; c) (C1-C6) alkyl, wherein (C1-C6) alkyl is substituted with one or more Z2 groups and optionally substituted with one or more Z1 groups; d) -X (C1-C6) alkyl, -X (C1-C6) haloalkyl, -X (C2-C6) alkenyl, -X (C2-C6) alkynyl and -X (C3-C7) carbocycle, wherein any -X (C1-C6) alkyl and -X (C1-C6) haloalkyl is substituted with one or more Z3 groups and |
| priorityDate | 2010-07-02-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 148.