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publicationNumber ES-2622953-T3
titleOfInvention Crystalline polymorph of a bisulfate salt of a thrombin receptor antagonist
abstract A process for the preparation of Compound 2 from Compound 1 according to the reaction: ** Formula ** comprising: d) mixing Compound 1 in acetonitrile to form a mixture; e) heat the mixture to a temperature of 50 ° C; and f) adding a mixture of sulfuric acid and acetonitrile to the heated mixture.
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