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filingDate 2010-08-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9c55d0ef58aec0d18e1c5d016025bf31
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publicationDate 2017-04-12-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2608670-T3
titleOfInvention 2- (Pyrimidin-5-yl) -thiopyrimidine derivatives as modulators of Hsp70 and Hsc70 for the treatment of proliferative disorders
abstract A compound of the formula 2a '** Formula ** or a stereoisomer, tautomer, or pharmaceutically acceptable salt thereof, wherein: each X and Y is independently selected from the group consisting of alkyl, alkenyl, or optionally straight or branched alkynyl replaced; an optionally substituted carbocyclic, heterocyclic, aryl, or heteroaryl group; halo; an optionally substituted C2-22acyl group; a group -NR4R5; a group -C (O) R6; a group - (ethoxy) n-R6, where n is 1-12; an optionally substituted alkoxycarbonyl group; an optionally substituted alkyloxy group; an optionally substituted amino group; a nitro group; and a carboxyl group; R4 and R5 are each independently selected from the group consisting of H; optionally substituted straight or branched alkyl, alkenyl, or alkynyl; and -C (O) R6; and each R6 is independently selected from the group consisting of an optionally substituted straight or branched alkyl, alkenyl, or alkynyl; an optionally substituted carbocyclic, heterocyclic, aryl, or heteroaryl group; an optionally substituted alkyloxy group; and an alkylacrylate group (such as ethyl acrylate).
priorityDate 2009-08-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036270
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374765
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68380742
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036140
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID70255
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID88960076
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036275
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374759
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419559184
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526579
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036157
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036276
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374760
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036158
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422531993
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036288
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID490325
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374761
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00764
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526573
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68380735
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036159
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID100135944
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP00775
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374762
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526574
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68380738
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036160
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID421033041
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036292
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374822
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036149
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422544112
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526584
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036284
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID692510
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68380751
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036152
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036285
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID3874950
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID68380753
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374818
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526587
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID6578
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374819
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526580
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036171
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID462188
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCP0DTC8
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID426374820
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526581
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036173
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID9257
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID122526582
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID156414
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID428036175

Total number of triples: 1921.