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filingDate 2013-01-22-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_abdfe9f4bc574d2b9f3f4298600ef3d8
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publicationDate 2017-03-17-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2605939-T3
titleOfInvention Integrin antagonist conjugates for administration directed to cells expressing alpha-V-beta-3
abstract A compound of formula I: ** Formula ** or a pharmaceutically acceptable salt or ester thereof; in which n is 1-24 and in which: R1 is selected from the group consisting of: (1) a compound of the formula: ** Formula ** in which m is 0 or 1; (2) a compound of the formula: ** Formula ** in which X is N or CH; (3) a compound of the formula: ** Formula ** (4) a compound of the formula: ** Formula ** (5) a compound of the formula: ** Formula ** R2 is selected from the group consisting in: (1) a compound of the formula: ** Formula ** (2) a compound of the formula: ** Formula ** (3) a compound of the formula: ** Formula ** and (4) a compound of the formula: ** Formula ** in which R3 is a conjugate moiety and X represents sulfur or a compound of the formula: ** Formula **
priorityDate 2012-01-27-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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