http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2602465-T3

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filingDate 2005-08-09-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2017-02-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_86429ff7833df4076e456c26693831ec
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1815f4cc041eaa4b9f0d397d38fb060b
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publicationDate 2017-02-21-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2602465-T3
titleOfInvention Combinations for the treatment of diseases that involve cell proliferation
abstract A pharmaceutical composition, comprising effective amounts of: (i) (A compound 1 of formula (I): ** Formula ** wherein the abbreviations X1, X2, X3, X4 and X5 used in the Table mean in each case a binding to the position in the general formula shown in the Table instead of the corresponding groups R1, R2, R3, R4 and L-R5, optionally in the form of their tautomers, racemates, enantiomers, diastereomers and mixtures thereof and optionally in the form of the pharmacologically acceptable acid, solvate, hydrate or polymorphic addition salts thereof; and (ii) at least one additional therapeutic agent 2 selected from the group consisting of vatalanib, gefitinib, erlotinib, iressa, tarceva, herceptin, atrasentan, rituximab, cetuximab, Avastin tm (bevacizumab), IMC-1C11, erbitux (C-225), DC-101, EMD-72000, vitaxin, imatinib, VEGFtrap, melphalan, cyclophosphamide, an oxazaphosphine, doxorubicamine (docloorubicamine) adriamycin), doxorubic ina liposomal (doxil), epirubicin, idarubicin, mitoxantrone, amsacrine, dactinomycin, distamycin, netropsin, pibenzimol, mitomycin, CC-1065, duocarmycin, mitramycin, chromomycin, olivomycin, propamidine, stilbamidine, an antramycin, an antramreacin phleomycin a bleomycin, liblomicina, navelbine, vinblastine, vincristine, vindesine, vinorelbine, colchicine, maytansine, fomopsina, dolastatin, etoposide, teniposide, combretastatin, anfetinilo, procarbazine, bortezomib, asparaginase, pegylated asparaginase (pegaspargase), inhibitor timidinafosforilasa, estramustine (T-66), megestrol, flutamide, casodex, anandron, cyproterone acetate, aminoglutethimide, anastrozole, formestan, letrozole, leuprorelin, buserelin, goserelin or triptorelin, tamoxifen, droloxifene, trioxifene, raloxifenoid, zindoxadiene, zindoxadiene, zindoxadiene, zindoxadiene finasteride, ketoconazole, leuprolide, prednisone, prednisolone, methylprednisolone, dexamethasone, budenoside, fluoc ortholone or triamcinolone, interferon, interferon β, IL-10, IL-12, etanercept, thalidomide, revimid mitomycin C, misonidazole, NLP-1 or NLA-1, nitromine, an anti-CD3 or anti-CD25 antibody, minodronic acid, Zoledronic acid monohydrate, ibandronate hydrated sodium, disodium clodronate, metronidazole, misonidazole, benznidazole, nimorazole, RSU-1069, SR-4233, bromodeoxyuridine, iododeoxyuridine, porphimer, photofrine, merocyanine 540 (MC-540, acetylpurine, acetylpurine acid, mesalazine, ibuprofen, naproxen, flurbiprofen, fenoprofen, fenbufen, ketoprofen, indoprofen, pirprofen, carprofen, oxaprozine, pranoprofen, miroprofen, thioxaprofen, suprofen, alminoprofen, thiaxaprofenocoenomethyl, toluprocophene, zupotophenochlorine, zuprocophene, zuprobenzene, zuprocophene, zuprobenzene, zuproenophenophenone , fenclofenac, alclofenac, bromfenac, ibufenac, aceclofenac, acemetacin, fentiazac, clidanac, etodolac, oxpinac, mefenamic acid, meclofenamic acid, flufenamic acid, acid Nifluminic, tolfenamic acid, diflunisal, flufenisal, piroxicam, tenoxicam, lornoxicam, nimesulide, meloxicam, celecoxib, rofecoxib, apolizumab, 1D09C3, TIMP-1, TIMP-2, Zinc, tetrathomolibdate, squattata, quantalatin, squattata, quantalatin, quantalatin, quantalatin, quantalatin, quantalatin, squat Neovastat, bicalutamide, abarelix, oregovomab, mitumomab, TLK-286, alemtuzumab, ibritumomab, temozolomide, denileukin diftitox, aldesleukin, dacarbazine, floxuridine, plicamycin, mitotane, pipobroman, or optionally, in combination with pharmaceutically, in combination with pharmaceutically, in combination with pharmaceutical acceptable, and optionally intended for co-treatment with radiotherapy or radio-immunotherapy, in the form of a combined preparation for simultaneous, separate or sequential use in the treatment of diseases involving cell proliferation, cell migration or apoptosis of cancer cells, or angiogenesis .
priorityDate 2004-08-14-04:00^^<http://www.w3.org/2001/XMLSchema#date>
type http://data.epo.org/linked-data/def/patent/Publication

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http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB1LEI7
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA4Y9A7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419504051
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCA3CZ93
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID41867
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419482154
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID415852
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419479716
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID410564866
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID776851
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCB0KPU9
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ31FE7
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID420277331
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID453991
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID419535646
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID16130954
http://rdf.ncbi.nlm.nih.gov/pubchem/protein/ACCQ8E927
http://rdf.ncbi.nlm.nih.gov/pubchem/gene/GID246266
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID22137869
http://rdf.ncbi.nlm.nih.gov/pubchem/compound/CID3080587
http://rdf.ncbi.nlm.nih.gov/pubchem/substance/SID422600813

Total number of triples: 919.