http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2586252-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_7c5e77c181522ee1fd44df1ae5ac2196 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-4365 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P35-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-048 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D495-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D513-04 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P35-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D513-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4355 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-437 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-4365 |
| filingDate | 2009-02-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2016-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9aea7add198266b888abe26e98042601 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1ae8759b708552a28e5b73f37512be05 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_048f664367f8735f54266c5e1b62176b http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_32e326ade08b12037b9c0076ad7c6afe |
| publicationDate | 2016-10-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2586252-T3 |
| titleOfInvention | Condensed heterocyclic derivative and use thereof |
| abstract | A compound represented by the formula ** Formula ** wherein X is O, S or N (C1-6 alkyl); R2 is (A) carbamoyl that optionally has 1 or 2 substituents that are selected from (1) C1-6 alkyl that optionally has 1 or 2 substituents that are selected from (1 ') halogen atom, (2') cyano, ( 3 ') amino, (4') C1-6 alkylamino, (5 ') di- C1-6 alkylamino optionally having a hydroxy, (6') C1-6 alkoxycarbonylamino, (7 ') hydroxy, (8' ) C1-6-alkyl-carbamoyl, (9 ') 5-7 membered cyclic carbamoyl, (10') heterocyclic group optionally possessing a (a) hydroxy, or (b) C1-5 alkyl optionally possessing a hydroxy , (11 ') C1-5 alkoxycarbonyl, and (12') C3-6 cycloalkyl, (2) C3-6 cycloalkyl optionally having 1 or 2 substituents selected from (1 ') amino, and (2' ) hydroxy, (3) C6-10 aryl, and (4) heterocyclic group optionally possessing a substituent that is selected from (1 ') C1-6 alkyl optionally possessing 1 or 2 substituents that are selected from (a) C6 aryl -10, and (b) hydroxy, (2 ') C 1-6 alkylcarbonyl optionally possessing a substituent selected from (a) C 1-6 alkylcarbonyloxy, and (b) hydroxy, (3 ') C 1-6 alkoxycarbonyl, and (4') 5- or 6-membered aromatic heterocyclic group, or (B) 5-7 membered cyclic carbamoyl optionally possessing a substituent that is selected from (1) C1-6 alkyl optionally possessing a substituent that is selected from (a) heterocyclic group, and (b) amino, (2) amino, ( 3) N-C 1-6 alkyl-N- (C 1-6 alkylcarbonyl) amino, (4) heterocyclic group, and (5) C 1-6 alkylcarbonyl optionally possessing a substituent selected from (a) hydroxy , (b) C1-6 alkoxy, (c) amino, and (d) C1-6 alkylamino; R3 is hydroxy optionally possessing (1) C1-6 alkyl optionally possessing a C1-6 alkoxy, or (2) C1-6 alkyl optionally possessing 1 to 3 halogen atoms; R4 is (1) hydrogen atom, or (2) C1-6 alkyl optionally possessing a substituent that is selected from (1 ') C3-6 cycloalkyl, (2') C6-10 aryl optionally possessing (i) 1 or 2 C1-6 alkoxy or (ii) 1 to 3 halogen atoms, (3 ') C1-6 alkylcarbonyl, (4') C6-10 carbonyl aryl optionally possessing a halogen atom or C1-6 alkoxy , (5 ') C1-6 alkoxycarbonyl, (6') C6-10 -carbamyl aryl, (7 ') heterocyclic group, (8') C6-10 aryloxy, and (9 ') carboxy; RA1 is a hydrogen atom or a C1-6 alkyl group; and RA2 is a hydrogen atom or a C1-6 alkyl group; or a salt thereof. |
| priorityDate | 2008-02-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 1806.