http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2582211-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_bb75b0b19820e3833ebdcb31603b242b |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-32 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D471-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D213-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D405-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-14 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D309-40 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D213-80 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D405-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D309-32 |
| filingDate | 2010-03-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2016-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_51e83f0940124ae59fdf919addb6fa9a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_f10e6eb05d943e31d73515faf9e77c5c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_14115e6208558c57f89577bd98c7b1dc http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_2b47106781a95555d35eebf320c0bf31 |
| publicationDate | 2016-09-09-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2582211-T3 |
| titleOfInvention | Process to produce pyrone and pyridone derivatives |
| abstract | A method of producing a compound shown by the formula (X4) or a salt thereof, comprising the steps of: reacting a compound shown by the formula (X2): ** Formula ** (in which R1d is hydrogen , halogen, C1-6 alkyloxy optionally substituted with substituent E, carbocyclyl C1-6 alkyloxy optionally substituted with substituent E, heterocyclyl C1-6 alkyloxy optionally substituted with substituent E, or -OSi (R1e) 3, the R1e are each independently alkyl C1-6 optionally substituted with substituent E, carbocyclyl optionally substituted with substituent E, heterocyclyl optionally substituted with substituent E, carbocyclyl C1-6 alkyl optionally substituted with substituent E or heterocyclyl C1-6 alkyl optionally substituted with substituent E, R2d is hydrogen, alkyl C1-6 optionally substituted with substituent E, carbocyclyl C1-6 alkyl optionally substituted with substituent E or heterocyclyl C1-6 alkyl optionally substituted with substituent E, R3d is hydrogen, C1-6 alkyl optionally substituted with substituent E, -N (R3e) 2 or -OR3e, the R3e are each independently C1-6 alkyl optionally substituted with substituent E or can be taken together to form a heterocycle and the wavy line is the E form and / or the Z form or the mixture thereof. Substituent E: halogen, cyano, hydroxy, carboxy, formyl, amino, oxo, nitro, C1-6 alkyl, halogen C1-6 alkyl, C1-6 alkyloxy, carbocyclyl optionally substituted with substituent F, heterocyclyl optionally substituted with substituent F, carbocyclyl C1-6 alkyloxy optionally substituted with substituent F, heterocyclyl C1-6 alkyloxy optionally substituted with substituent F, carbocyclyl C1-6 alkylthio optionally substituted with substituent F, heterocyclyl C1-6 alkylthio optionally substituted with substituent F, carbocyclyl C1-6 alkylamino optionally substituted with substituent F, heterocyclyl C1-6 alkylamino optionally substituted with substituent F, carbocyclyloxy optionally substituted with substituent F, heterocyclyloxy optionally substituted with substituent F, carbocyclylcarbonyl optionally substituted with substituent F, heterocyclylcarbonyl optionally substituted with substituent F, carbocyclylaminocarbonyl substituted with s usstituent F, heterocyclylaminocarbonyl optionally substituted with substituent F, halogen C1-6 alkyloxy, C1-6 alkyloxy C1-6 alkyl, C1-6 alkyloxy C1-6 alkyloxycarbonyl C1-6, alkyloxycarbonyl C1-6, alkyloxycarbonylamino C1-6, alkylamino C1-6, C1-6 alkylcarbonylamino, C1-6 alkylaminocarbonyl, C1-6 alkylsulfonyl and C1-6 alkylsulfonylamino; Substituent F: halogen, hydroxy, carboxy, amino, oxo, nitro, C1-6 alkyl, halogen C1-6 alkyl, C1-6 alkyloxy and amino protecting group). with a compound shown by the formula (V2): ** Formula ** (wherein R4d is C1-6 alkyl optionally substituted with substituent E, carbocyclyl C1-6 alkyl optionally substituted with substituent E or heterocyclyl C1-6 alkyl optionally substituted with substituent E, R5d is hydrogen, halogen, C1-6 alkyloxy optionally substituted with substituent E, or -O-SO2-R5e, R5e is C1-6 alkyl optionally substituted with substituent E, carbocyclyl optionally substituted with substituent E, optionally substituted heterocyclyl with substituent E, carbocyclyl C1-6 alkyl optionally substituted with substituent E or heterocyclyl C1-6 alkyl optionally substituted with substituent E and substituent E defined above) to obtain a compound shown by the formula (X3): ** Formula * * (in which each symbol has been defined above); and reacting the compound shown by the formula (X3) with a compound shown by the formula (V3): ** Formula ** (wherein R6d is optionally substituted C1-6 alkyl with substituent E, optionally substituted C1-6 alkenyl with substituent E, amino optionally substituted with substituent E, C1-6 alkylamino optionally substituted with substituent E, carbocyclyl optionally substituted with substituent E or heterocyclyl optionally substituted with substituent E and substituent E defined above) to obtain a compound shown by the formula (X4): ** Formula ** (in which each symbol has been defined above). |
| priorityDate | 2009-03-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 397.