http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2569511-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_f2d3599fb8f8f479dba95ca9bb504884 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-06 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P7-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D491-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D498-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P17-02 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P21-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P19-00 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-537 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P29-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D491-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D498-10 |
| filingDate | 2008-11-13-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2016-05-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_feb6d8c57fb549a0d32f456381f5d1c1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1dbb91d7e2f495e30905c571a53f2643 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_0e253017786cac135cdd49e6fc069738 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_23392f7d5a16cdbe7357d9404783144a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b341efb769de74e7b27b0259731d858c |
| publicationDate | 2016-05-11-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2569511-T3 |
| titleOfInvention | ENT1 Nucleoside Balancing Conveyor Inhibitors |
| abstract | Compound of formula (1) ** Formula ** including any stereochemically isomeric form thereof, in which -A-B- represents ** Formula ** in which n is an integer 0 or 1; R13 represents hydroxy or halo; R14 represents hydrogen or C1-6 alkyl; in the bivalent radicals (a-4), (a-5) and (a-6), any of the hydrogen atoms in the same or in a different carbon atom may be substituted by halo; R1 and R2 are each independently selected from hydrogen, halo or C1-6 alkyl; R3, R4, R5 and R6 are each independently selected from hydrogen, halo, C1-6 alkyl, polyhalo-C1-6 alkyl, C3-6 cycloalkyl, NO2, Cycle1, Cycle2, or X-R8, in the that X represents O or NR9, in which R9 is hydrogen, C1-6 alkyl or C1-6 alkyl-oxy C1-6 alkyl, and in which R8 is hydrogen, C1-6 alkyl, C2 alkenyl -6, C3-6 cycloalkyl, polyhalo-C1-6 alkyl, C1-6 alkyl oxycarbonyl, C1-6 alkylcarbonyl, polyhalo-C1-6 alkylcarbonyl, Cycle2, - (C> = O) - (CH2) m-Cycle2, - (C> = O) - (CH2) m-CH2-OH, - (C> = O) - (CH2) m-CH2-O-C1-4 alkyl or C1 alkyl -6 substituted with halo, hydroxy, cyano, C3-6 cycloalkyl, C1-6-oxy alkyl, aminocarbonyl, phenyl, Cycle1, or Cycle2, or NR11R12, wherein R11 and R12 are each independently selected from hydrogen, alkyl C1-6, C1-6 alkylcarbonyl, or C1-6 alkyl oxycarbonyl; m is an integer of 0, 1 or 2; Cycle 1 is selected from ** Formula ** in which R 10 is hydrogen, C 1-6 alkyl, C 1-6 alkylcarbonyl, or C 1-6 alkyl oxycarbonyl; and Cycle2 is selected from where R10 is hydrogen, C1-6 alkyl, C1-6 alkylcarbonyl, C1-6 alkylcarboxylic or C1-6alkyl substituted by halo or hydroxy; or a pharmaceutically acceptable acid addition salt thereof, or a solvate thereof, or an N-oxide form thereof. |
| priorityDate | 2007-11-14-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
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