http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2553246-T3
Outgoing Links
| Predicate | Object |
|---|---|
| assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_966a6c1f382ec9bcb5e3839dfd73e5b8 |
| classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P5-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-20 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P25-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P1-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61K31-5517 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P15-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P9-12 |
| classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P15-10 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P1-16 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D487-04 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D519-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61K31-5517 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-22 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-24 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P25-18 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P13-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A61P9-04 |
| filingDate | 2011-04-21-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| grantDate | 2015-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3fa292408c19a9787409f0a5c3d7ff9e http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_9f811184bcd368b898cfc7aaf03ea193 |
| publicationDate | 2015-12-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| publicationNumber | ES-2553246-T3 |
| titleOfInvention | Heterobiaryl-cyclohexyl-tetraazabenzo [e] azulenes |
| abstract | A compound of the formula I ** Formula ** in which R1 is selected from the group consisting of: i) H, ii) -C1-6 alkyl, unsubstituted or substituted 1 to 5 times by substituents individually selected from the group consisting of OH, halogen, cyano and C1-6 alkoxy, iii) -S (O) 2-C1-6 alkyl, whose C1-6 alkyl is unsubstituted or substituted 1 to 5 times by substituents individually selected from the group formed by OH, halogen, cyano and C1-6 alkoxy, iv) -C (O) -C1-6 alkyl, whose C1-6 alkyl is unsubstituted or substituted 1 to 5 times by substituents individually selected from the group consisting of OH, halogen, cyano and C1-6 alkoxy, v) -C (O) O-C1-6 alkyl, whose C1-6 alkyl is unsubstituted or substituted 1 to 5 times by substituents individually selected from the group consisting of OH , halogen, cyano and C1-6 alkoxy; vi) cycloalkyl, unsubstituted or substituted 1 to 5 times by substituents individually selected from the group consisting of OH, halogen, cyano, C1-6 alkyl and C1-6 alkoxy, vii) S (O) 2- (CH2) q -NRiRii, in which q is the number 0 or 1, Ri and Rii independently of each other are chosen from the group consisting of H and C1-6 alkyl, or Ri and Rii together with the nitrogen to which they are attached form a heterocyclyl from 3 to 7 links containing one or two heteroatoms chosen individually from N, O and S, and said heterocyclyl is unsubstituted or substituted 1 to 5 times by substituents individually selected from the group consisting of oxo, halogen, C1-6 alkyl and C1-6 alkoxy, viii) - (CH2) r-NRiiiRiv, in which r is the number 1, 2 or 3, Riii and Riv independently from each other are chosen from the group consisting of H and C1-6 alkyl, or Riii and Riv together with the nitrogen to which they are attached form a heterocyclyl of 3 to 7 links containing one or two heteroatoms chosen individually. id. N, O and S, and said heterocyclyl is unsubstituted or substituted 1 to 5 times by substituents individually selected from the group consisting of oxo, halogen, C1-6 alkyl and C1-6 alkoxy, and ix) -C ( O) (CH2) s-NRvRvi, in which s is the number 1, 2 or 3, Rv and Rvi independently of each other are chosen from the group consisting of H and C1-6 alkyl, or Rv and Rvi together with the nitrogen to which they are attached form a heterocyclyl of 3 to 7 links containing one or two heteroatoms chosen individually from N, O and S, and said heterocyclyl is unsubstituted or substituted 1 to 5 times by substituents chosen individually from the group consisting of oxo, halogen, C1-6 alkyl and C1-6 alkoxy; R2 is halogen; R3 is heterobaryl, unsubstituted or substituted by 1-5 substituents individually selected from the group consisting of OH, halogen, cyano, C1-6 alkyl, C1-6 alkoxy, halogen-C1-6 alkyl, halogen-C1-6 alkoxy e hydroxyC 1-6 alkyl; or a pharmaceutically acceptable salt thereof. |
| priorityDate | 2010-04-26-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
| type | http://data.epo.org/linked-data/def/patent/Publication |
Incoming Links
Total number of triples: 124.