http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2552097-T3
Outgoing Links
Predicate | Object |
---|---|
assignee | http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_648c9679dd9ec36125406a2dafa6bf7e |
classificationCPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D239-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D239-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A01N47-38 |
classificationIPCInventive | http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N43-54 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/A01N47-38 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D401-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D409-12 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-47 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D239-46 |
filingDate | 2010-08-05-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate | 2015-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor | http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_361370bcb91f0fa6e237548a4f5a2e8d http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_81782f78a9e26159d7ef8c6cac2c7cd1 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_8c106873c6fee4c88d39b9ec8a2a26f5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a4649a70056a96f07e288ab9f8e9a921 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_3b0a955303a2fcdcd7284f522d3dbcd5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1c63780dd745a76941ea7f285cb3eee5 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_de605d25eb9401c45648bf2cf7403a1a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_ad79e56dc08b409c085b57ffd679949c http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5d6e08a2afcb00cda11cba3c35425352 |
publicationDate | 2015-11-25-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber | ES-2552097-T3 |
titleOfInvention | 5-Fluoro-2-oxopyrimidinone-1 (2H) -carboxamide derivatives substituted in N1 |
abstract | A compound according to Formula I: ** Formula ** wherein R1 is: H; C1-C6 alkyl optionally substituted by 1-3 R4; C1-C6 alkenyl optionally substituted by 1-3 R4; C3-C6 alkynyl optionally substituted by 1-3 R4; phenyl or benzyl, wherein each of phenyl or benzyl may optionally be substituted with 1-3 R5, or with a 5-6 membered saturated or unsaturated ring system, or with a 5-6 membered fused ring system, or with a system of fused rings of 6-6 members, each containing 1-3 heteroatoms where each ring can be optionally substituted by 1-3 R5, biphenyl or naphthyl optionally substituted by 1-3 R5; - (CHR6) mOR7; -C (> = O) R8; -C (> = S) R8; -C (> = O) OR8; -C (> = S) OR8; - (CHR6) m N (R9) R10; -C (> = O) N (R9) R10; or -C (> = S) N (R9) R10; where m is an integer from 1 to 3; R2 is H or C1-C6 alkyl optionally substituted by R4; Alternatively, R1 and R2 can be taken together to form> = CR11N (R12) R13; R3 is -C (> = O) N (R9) R10 or -C (> = S) N (R9) R10; R4 is independently halogen, C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxy, C1-C6 haloalkoxy, C1-C4 alkylthio, C1-C4 haloalkylthio, halotium, amino, C1-C3 alkylamino, C2-C6 alkoxycarbonyl, alkylcarbonyl C2-C6, C2-C6 alkylaminocarbonyl, hydroxyl, or C3-C6 trialkylsilyl; R5 is independently halogen, C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxy, C1-C6 haloalkoxy, C1-C6 alkylthio, C1-C6 haloalkylthio, halotium, amino, C1-C6 alkylamino, C2-C6 dialkylamino, alkoxycarbonyl C2-C6, or C2-C6 alkylcarbonyl, nitro, hydroxyl, or cyano; R6 is H, C1-C6 alkyl, C1-C6 alkoxy, benzyl or phenyl, wherein each of benzyl or phenyl may optionally be substituted with 1-3 R5; R7 is H, C1-C6 alkyl, C2-C6 alkenyl, C3-C6 alkynyl, C1-C6 haloalkyl, C1-C6 alkoxyalkyl, C2-C6 alkylcarbonyl, phenyl or benzyl, wherein each of benzyl or phenyl can optionally be substituted for 1-3 R5, or with a system of saturated or unsaturated rings of 5-6 members, or with a system of fused rings of 5-6 members, or with a system of fused rings of 6-6 members, containing each 1-3 heteroatoms where each ring can be optionally substituted by 1-3 R5, biphenyl or naphthyl optionally substituted by 1-3 R5; R8 is H, C1-C6 alkyl, C2-C6 alkenyl, C3-C6 alkynyl, C1-C6 haloalkyl, C1-C6 alkoxyalkyl, phenyl or benzyl, wherein each of phenyl or benzyl may optionally be substituted with 1-3 R5 , or with a system of saturated or unsaturated rings of 5-6 members, or with a system of fused rings of 5-6 members, or with a system of fused rings of 6-6 members, each containing 1-3 heteroatoms in where each ring can be optionally substituted by 1-3 R5, biphenyl or naphthyl optionally substituted by 1-3 R5; R9 is H, C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyalkyl, C1-C6 alkylalkoxycarbonyl, C2-C6 alkylcarbonyl, - (CH2) mSCH3, phenyl or benzyl, wherein each of phenyl or benzyl can be substituted optionally for 1-3 R5, or for a system of saturated or unsaturated rings of 5-6 members, or with a system of fused rings of 5-6 members, or with a system of fused rings of 6-6 members, each containing one 1-3 heteroatoms where each ring can be optionally substituted by 1-3 R5, biphenyl or naphthyl optionally substituted by 1-3 R5, R10 is H, C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyalkyl, alkylcarbonyl C2-C6, benzyl, wherein the benzyl can be optionally substituted with 1-3 R5; alternatively R9 and R10 can be taken together to form a saturated or unsaturated 5-6 membered ring containing 1-3 heteroatoms, where each ring can be optionally substituted with 1-3 R5; R11 is H or C1-C4 alkyl; R12 is H, cyano, hydroxyl, C1-C4 alkyl, C1-C6 alkoxy, C2-C6 alkylcarbonyl, phenyl or benzyl, wherein each of phenyl or benzyl, may optionally be substituted with 1-3 R5; or by a system of saturated or unsaturated rings of 5-6 members, or by a system of fused rings of 5-6 members, or by a system of fused rings of 6-6 members, each containing 1-3 hetero atoms where each ring may optionally be substituted with 1-3 R5, biphenyl or naphthyl optionally substituted with 1-3 R5; alternatively R11 and R12 can be taken together to form a saturated or unsaturated 5-6 membered ring containing 1-3 heteroatoms, where each ring can be optionally substituted with 1-3 R5; R13 is H, C1-C4 alkyl, C1-C6 alkoxy, C2-C6 alkylcarbonyl, phenyl or benzyl, wherein each phenyl or benzyl can optionally be substituted with 1-3 R5; and alternatively R12 and R13 can be taken together to form a saturated or unsaturated 5-6 membered ring containing 1-3 heteroatoms, where each ring can be optionally substituted with 1-3 R5, |
priorityDate | 2009-08-07-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type | http://data.epo.org/linked-data/def/patent/Publication |
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Total number of triples: 1702.