http://rdf.ncbi.nlm.nih.gov/pubchem/patent/ES-2533026-T3

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filingDate 2011-06-01-04:00^^<http://www.w3.org/2001/XMLSchema#date>
grantDate 2015-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
inventor http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_936ab4ded3a64dda28add4d86f8dc53b
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publicationDate 2015-04-07-04:00^^<http://www.w3.org/2001/XMLSchema#date>
publicationNumber ES-2533026-T3
titleOfInvention N - [(het) arylalkyl)] pyrazole (thio) carboxamides and their hetero substituted analogs
abstract A compound of formula (I): ** Formula ** in which - X1 and X2, which may be the same or different, represent a halogen atom; - Y represents a C1-C4 alkyl; - T represents O or S; - W represents CZ4Z5; OR; S; SW; SO2; NZ6; SiZ7Z8; or -C (> = U) -; - B represents a phenyl ring that may be substituted by up to 5 X groups that may be the same or different; a naphthyl ring that may be substituted by up to 7 X groups that may be the same or different; or a saturated, partially saturated or unsaturated, monocyclic or bicyclic fused ring of 4, 5, 6, 7, 8, 9, 10 members comprising 1 to 4 heteroatoms selected from the list consisting of N, O, S, which it can be substituted by up to 6 X groups that can be the same or different; -X represents a halogen atom; nitro; cyano; isonitrile; hydroxy; Not me; sulfanyl; pentafluoro-λ6-sulfanyl; formyl; formyloxy; formylamino; a substituted or unsubstituted (hydroxy-imino) -C 1 -C 8 alkyl group; (C1-C8 alkoxy-imino) -C1-C8 alkyl; (C2-C8 alkenyloxy-imino) -C1-C8 substituted or unsubstituted alkyl; (C2-C8 alkynyloxy-imino) -C1-C8 substituted or unsubstituted alkyl; (benzyloxy-imino) -C1-C8 substituted or unsubstituted alkyl; carboxy; carbamoyl; N-hydroxycarbamoyl; carbamate; C1-C8 substituted or unsubstituted alkyl; C1-C8 halogenoalkyl having 1 to 5 halogen atoms; C2-C8 substituted or unsubstituted alkenyl; C2-C8 halogenoalkenyl having 1 to 5 halogen atoms; C2-C8 substituted or unsubstituted alkynyl; C2-C8 halogenoalkynyl having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkoxy; C1-C8 halogenoalkoxy having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkylsulfanyl; C1-C8 halogenoalkoxysulfanyl having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkylsulfinyl; C1-C8 halogenoalquisulfinyl having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkylsulfonyl; C1-C8 halogenoalquisulfonyl having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkylamino; C1-C8 substituted or unsubstituted dialkylamino; C2-C8 substituted or unsubstituted alkenyloxy; C2-C8 halogenoalkenyloxy having 1 to 5 halogen atoms; C3-C8 substituted or unsubstituted alkynyloxy; C2-C8 halogenoalkyloxy having 1 to 5 halogen atoms; C3-C7 substituted or unsubstituted cycloalkyl; C3-C7 halogenocycloalkyl having 1 to 5 halogen atoms; (C3-C7 cycloalkyl) -C1-C8 substituted or unsubstituted alkyl; (C3-C7 cycloalkyl) -C2-C8 substituted or unsubstituted alkenyl; (C3-C7 cycloalkyl) -C2-C8 substituted or unsubstituted alkynyl; tri (C1-C8 alkyl) substituted or unsubstituted; tri (C1-C8 alkyl) silyl substituted or unsubstituted C1-C8 alkyl; C1-C8 substituted or unsubstituted alkylcarbonyl; C1-C8 halogenoalkylcarbonyl having 1 to 5 halogen atoms; C1-C8 alkyl substituted or unsubstituted carbonyloxy; C1-C8 halogenoalkylcarbonyloxy having 1 to 5 halogen atoms; C1-C8 alkyl substituted or unsubstituted carbonylamino; C1-C8 halogenoalkylcarbonylamino having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkoxycarbonyl; C1-C8 halogenoalkyl carbonyl having 1 to 5 halogen atoms; C1-C8 alkyloxy substituted or unsubstituted; C1-C8 halogenoalkoxycarbonyloxy having 1 to 5 halogen atoms; C1-C8 alkyl substituted or unsubstituted carbamoyl; dialkyl C1-C8 substituted or unsubstituted carbamoyl; C1-C8 alkylamino substituted or unsubstituted; C1-C8 substituted or unsubstituted dialkylamino; N- (C1-C8-alkyl) hydroxy carbamoyl; C1-C8 alkoxy substituted or unsubstituted carbamoyl; N- (C1-C8 alkyl) - C1-C8 alkoxy-carbamoyl; aryl that may be substituted by up to 6 Q groups that may be the same or different; C1-C8 arylalkyl which may be substituted by up to 6 Q groups that may be the same or different; C2-C8 arylalkenyl which may be substituted by up to 6 Q groups that may be the same or different; C2-C8 arylalkyl which may be substituted by up to 6 Q groups that may be the same or different; aryloxy which may be substituted by up to 6 Q groups that may be the same or different; arylsulfanyl which may be substituted by up to 6 Q groups that may be the same or different; arylamino, which may be substituted by up to 6 Q groups that may be the same or different; C1-C8 arylakyloxy which may be substituted by up to 6 Q groups that may be the same or different; C 1 -C 8 arylalkyl sulfanyl, which may be substituted by up to 6 Q groups that may be the same or different; C 1 -C 8 arylalkyl amino, which may be substituted by up to 6 Q groups that may be the same or different; or - two substituents X together with the consecutive carbon atoms to which they are attached may form a 5 or 6 membered ring, saturated carbocycle or saturated heterocycle, which may be substituted by up to four Q groups that may be the same or different; - Z1 represents a hydrogen atom; a formyl group; a substituted or unsubstituted C1-C8 alkyl; C1-C8 substituted or unsubstituted alkoxy; C3-C7 cycloalkyl or a C3-C7 cycloalkyl substituted by up to 10 atoms or groups that may be the same or different and that may be selected from the list consisting of halogen, cyano, C1-C8 alkyl, C1-C8 halogenoalkyl atoms which It comprises up to 9 halogen atoms that can be the same or different, C1-C8 alkoxy, C1-C8 halogenoalkoxy comprising up to 9 halogen atoms that can be the same or different, C1-C8 alkoxycarbonyl, C1-C8 halogenoalkoxy carbonyl comprising up to 9 halogen atoms that may be the same or different, C1-C8-alkylaminocarbonyl or C1-C8-dialkylaminocarbonyl; - Z2, Z3, Z4 and Z5 independently represent a hydrogen atom; a halogen atom, cyano; C1-C8 alkyl substituted or unsubstituted C1-C8 halogenoalkyl having 1 to 5 halogen atoms; C1-C8 substituted or unsubstituted alkoxy; C1-C8 substituted or unsubstituted alkylsulfanyl; or C1-C8 substituted or unsubstituted alkoxy; or two substituents Zi and Zi + 1 being i an integer between 2 and 4, together with the consecutive carbon atoms to which they are attached can form a saturated carbocycle of 3, 4, 5, or 6 or 7 members that can be substituted by up to four groups that may be the same or different and that may be selected from the list consisting of halogen atoms, C1-C8 alkyl or C1-C2 halogenoalkyl comprising up to 5 halogen atoms that may be the same or different; - Z6 represents a hydrogen atom; a substituted or unsubstituted C1-C8 alkyl; a C1-C8 halogenoalkyl comprising up to 9 halogen atoms that may be the same or different; a substituted or unsubstituted C2-C8 alkenyl; a C2-C8 halogenoalkyl comprising up to 9 halogen atoms that may be the same or different; a substituted or unsubstituted C3-C8 alkynyl; a C3-C8 halogenoalkyl comprising up to 9 halogen atoms that may be the same or different; a substituted or unsubstituted C3-C7 cycloalkyl; a C3-C7 halocyclocycloalkyl comprising up to 9 halogen atoms that may be the same or different; a C3-C7 cycloalkyl-substituted or unsubstituted C1-C8 alkyl; formyl; C1-C8 alkyl substituted or unsubstituted; a C1-C8 halogenoalkylcarbonyl comprising up to 9 halogen atoms that may be the same or different, a substituted or unsubstituted C1-C8 alkoxy; a C1-C8 halogenoalkoxycarbonyl comprising up to 9 halogen atoms that may be the same or different; a substituted or unsubstituted C1-C8 alkylsulfonyl; a C1-C8 halogenoalkylsulfonyl comprising up to 9 halogen atoms that may be the same or different; phenylmethylene which may be substituted by up to 7 Q groups that may be the same or different; or phenylsulfonyl which may be substituted by up to 5 Q groups that may be the same or different; - Z7 and Z8 independently represent a substituted or unsubstituted C1-C8 alkyl; - U represents O; S; N-ORa; or N-CN; - Ra represents a hydrogen atom; a substituted or unsubstituted C1-C4 alkyl; or a C1-C4 halogenoalkyl comprising up to 7 halogen atoms that may be the same or different; -Q independently represents a halogen atom; cyano; nitro; C1-C8 substituted or unsubstituted alkyl; C1-C8 halogenoalkyl having 1 to 9 halogen atoms that may be the same or different; C1-C8 substituted or unsubstituted alkoxy; C1-C8 halogenoalkoxy having 1 to 9 halogen atoms that may be the same or different, substituted or unsubstituted C1-C8 alkylsulfanyl; C1-C8 halogenoalkylsulfanyl having 1 to 9 halogen atoms that may be the same or different, substituted or unsubstituted tri (C1-C8 alkyl) silyl; substituted or unsubstituted C1-C8 trialkyl (C1-C8) alkyl; (C1-C8 alkoxy-imino) -C1-C8 substituted or unsubstituted alkyl; (benzyloxyimino) -C1-C8 alkyl; as well as its salts, N-oxides, metal complexes, metalloid complexes and optically active isomers.
priorityDate 2010-06-03-04:00^^<http://www.w3.org/2001/XMLSchema#date>
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Total number of triples: 1355.