Predicate |
Object |
assignee |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentassignee/MD5_ad7db51775730aa88bfb46e8c6b4ab71 |
classificationCPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/A61P43-00 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-416 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-404 http://rdf.ncbi.nlm.nih.gov/pubchem/patentcpc/C07D207-46 |
classificationIPCInventive |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-40 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-404 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-46 http://rdf.ncbi.nlm.nih.gov/pubchem/patentipc/C07D207-416 |
filingDate |
2004-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
grantDate |
2013-05-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
inventor |
http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1a6c520394c494ce3c05712550e2314a http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_1be11ec72f12ca1870207629cfd63e1d http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_55b94456e4115d0a2eee8d7426c3d7fd http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_c1c83b9fba5057a37b8e3197217c9aaf http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_7051557751ca55404ef2d934d5607589 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_b0c7d6bd71cb4cdc52d0892963f4b2f2 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_089b36e376201482007dbe18b9566786 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_939ff5e65e12197cab604a01be98a820 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_a48052781fbc662e85bcc750c2d406c9 http://rdf.ncbi.nlm.nih.gov/pubchem/patentinventor/MD5_5b66fdd1a4e88c3afe16d1b7f8043541 |
publicationDate |
2013-05-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
publicationNumber |
ES-2405329-T3 |
titleOfInvention |
Synthesis of acyloxyalkyl carbonate prodrugs and intermediates thereof |
abstract |
A process for synthesizing a 1- (acyloxy) -alkyl and Nhydrosuccinimidyl carbonate compound of formula (I), comprising: ** Formula ** (i) contacting a compound of formula (IV) and a compound of formula ( V) to provide a compound of formula (VI); (ii) contacting the compound of formula (VI) with a carboxylate compound of formula (VII) to provide an acyloxyalkyl thiocarbonate compound of formula (VIII); and (iii) contacting the thiocarbonate compound of formula (VIII) with an oxidant (IX), in the presence of an N-hydroxysuccinimide compound of formula (X) to provide the compound of formula (I): ** Formula ** |
priorityDate |
2003-12-30-04:00^^<http://www.w3.org/2001/XMLSchema#date> |
type |
http://data.epo.org/linked-data/def/patent/Publication |