| abstract |
Compounds selected from group No. Name and / or structure "A1" 6- (1-Methyl-1H-pyrazol-4-yl) -2- {3- [5- (2-morpholin-4-yl-ethoxy) -pyrimidin-2-yl] -benzyl} -2H-pyridazin-3-one, sulfate "A2" 6- (1-Methyl-1H-pyrazol-4-yl) -2- {3- [5- (2-morpholin-4-yl-ethoxy ) -pyrimidin-2-yl] -benzyl} -2H-pyridazin-3-one, mesylate "A3" 6- (1-Methyl-1H-pyrazol-4-yl) -2- {3- [5- (2 -morpholin-4-yl-ethoxy) -pyrimidin-2-yl] -benzyl} -2H-pyridazin-3-one, besylate "A4" 6- (1-Methyl-1H-pyrazol-4-yl) -2- {3- [5- (2-Morpholin-4-yl-ethoxy) -pyrimidin-2-yl] -benzyl} -2H-pyridazin-3-one, p-tosylate "A5" 6- (1 Methyl-1H-pyrazole -4-yl) -2- {3- [5- (2-morpholin-4-yl-ethoxy) -pyrimidin-2-yl] -benzyl} -2H-pyridazin-3-one, fumarate "A6" 6- (1-Methyl-1H-pyrazol-4-yl) -2- {3- [5- (2-morpholin-4-yl-ethoxy) pyrimidin-2-yl] -benzyl} -2H-pyridazin-3-one , "A7" maleate 3- (1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy) pyrimidin-2-yl] -benzyl} -6-oxo-1,6-dihydro-pyridazin-3 -yl) -benzonitrile, hydrochloride monohydrate "A8" 3- (1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy) -pyrimidin-2-yl] -benzyl} -6-oxo-1, 6-dihydro-pyridazin-3-yl) -benzonitrile, hydrobromide "A9" 3- ( 1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy) -pyrimidin-2-yl] -benzyl} -6-oxo-1,6-dihydro-pyridazin-3-yl) -benzonitrile, mesylate "A10" 3- (1- {3- [5- (1-Methyl-pipeddin-4-ylmethoxy) -pyrimidin-2-yl] -benzyl} -6-oxo-1,6-dihydro-pyridazin-3- il) -benzonitrile, besylate "A11" 3- (1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy) -pyrimidin-2-yl] -benzyl} -6-oxo-1,6- dihydro-pyridazin-3-yl) -benzonitrile, malate "A12" 3- (1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy) -pyrimidin-2-yl] -benzyl} -6- oxo-1,6-dihydro-pyridazin-3-yl) -benzonitrile, fumarate "A13" 3- (1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy) -pyrimidin-2-yl] -benzyl} -6-oxo-1,6-dihydro-pyridazin-3-yl) -benzonitrile, maleate "A14" 3- (1- {3- [5- (1-Methyl-piperidin-4-ylmethoxy)) - pyrimidin-2-yl] -benzyl} -6-oxo-1,6-dihydro-pyridazin-3-yl) -benzonitrile, p-tosylate, as well as their tautomers and stereoisomers, including mixtures thereof in all proportions. |